SCHEMBL7766546

SCHEMBL7766546

NS(=O)(=O)c1ccc(-c2ccc(OC[C@H](O)CCc3cccnc3)cc2)cc1F

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ADAMTS4 O75173 1/20 0.37
ADRB1 P08588 3/20 0.37
ADRB3 P13945 3/20 0.37
NAMPT P43490 1/20 0.37
ALDH1A1 P00352 1/20 0.36
ADRB2 P07550 2/20 0.36
PTAFR P25105 2/20 0.36
MMP12 P39900 1/20 0.36
FFAR1 O14842 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
F10 P00742 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7766538 1.00 CYP3A4 (0.39) CYP3A4MEN1KMT2AADAMTS4ADRB1
SCHEMBL7769942 0.90 MEN1 (0.39) CYP3A4MEN1KMT2AADAMTS4ADRB1
SCHEMBL7769940 0.90 MEN1 (0.39) CYP3A4MEN1KMT2AADAMTS4ADRB1
SCHEMBL7769952 0.89 GYS1 (0.38) MEN1KMT2AADAMTS4ADRB1ADRB3
SCHEMBL7769949 0.89 GYS1 (0.38) MEN1KMT2AADAMTS4ADRB1ADRB3
SCHEMBL7976666 0.85 CYP3A4 (0.39) CYP3A4ADAMTS4NAMPTPTAFR
SCHEMBL7976671 0.85 CYP3A4 (0.39) CYP3A4ADAMTS4NAMPTPTAFR
SCHEMBL4853590 0.85 CA2 (0.50) MEN1KMT2AADAMTS4ADRB1ADRB3
SCHEMBL7771595 0.85 CA2 (0.50) MEN1KMT2AADAMTS4ADRB1ADRB3
SCHEMBL7772401 0.84 MEN1 (0.40) CYP3A4MEN1KMT2AADAMTS4ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115706-A1 NOVEL COMPOUNDS AstraZeneca AB (SE) 2001-07-18 EP claimed
WO-2000018730-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2000-04-06 WO claimed
EP-1115706-A1 NOVEL COMPOUNDS AstraZeneca AB (SE) 2001-07-18 EP disclosed
WO-2000018730-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2000-04-06 WO disclosed