SCHEMBL7767780

SCHEMBL7767780

O=C1C(=CO)Cc2ccc(F)cc21

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.49
MAOB P27338 4/20 0.49
CES2 O00748 4/20 0.46
TNF P01375 2/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
ACHE P22303 1/20 0.40
PARP1 P09874 1/20 0.40
PARP10 Q53GL7 1/20 0.40
LCK P06239 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7767777 1.00 MAOA (0.49) MAOAMAOBCES2TNFCA1
SCHEMBL12819448 0.85 PARP1 (0.46) MAOAMAOBCA1CA2CA7
SCHEMBL12965293 0.85 PARP1 (0.46) MAOAMAOBCA1CA2CA7
SCHEMBL7767503 0.79 METAP1 (0.57) MAOAMAOBCES2TNFCA1
SCHEMBL7767505 0.79 METAP1 (0.57) MAOAMAOBCES2TNFCA1
SCHEMBL26073771 0.76 BCHE (0.52) MAOAMAOBCA1CA2CA7
SCHEMBL4808970 0.76 MIF (0.61) MAOAMAOBCES2ACHE
SCHEMBL4808965 0.76 MIF (0.61) MAOAMAOBCES2ACHE
SCHEMBL21801661 0.75 CES2 (0.46) MAOAMAOBCES2LCK
SCHEMBL11428273 0.74 MIF (0.62) MAOAMAOBTNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700905-B1 Tricyclic pyrazole derivatives HOFFMANN LA ROCHE (CH) 2001-10-31 EP disclosed
US-5561150-A 1-AMINOALKYL-1,4-DIHYDROINDENO(2,1-C)PYRAZOLES OR 1H-BENZ(G)INDAZOLES; SEROTONIN RECEPTOR ANTAGONISTS; ANTIDEPRESSANTS; NERVOUS SYSTEM, PSYCHOLOGICAL AND GASTROINTESTINAL DISORDERS HOFFMAN-LA ROCHE INC. (US) 1996-10-01 US disclosed
EP-0700905-A1 Tricyclic pyrazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1996-03-13 EP disclosed