SCHEMBL7769189

SCHEMBL7769189

CC(C)COc1nc(O)cc(C(F)(F)F)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.40
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
PTGS2 P35354 6/20 0.34
PTGS1 P23219 4/20 0.34
CYP2C19 P33261 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
CRHBP P24387 1/20 0.34
CRHR2 Q13324 1/20 0.34
HSD17B10 Q99714 1/20 0.34
XDH P47989 1/20 0.33
LMNA P02545 1/20 0.33
SYK P43405 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
PDK2 Q15119 1/20 0.32
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7769381 0.79 PTGS2 (0.46) RXRARXRBPTGS2PTGS1HSD17B10
SCHEMBL5998545 0.79 PTGS1 (0.51) RXRARXRBTLR7PTGS2PTGS1
SCHEMBL601281 0.76 HSD17B10 (0.54) RXRARXRBPTGS2PTGS1HSD17B10
SCHEMBL7457755 0.72 TLR7 (0.38) TLR7PTGS2CYP2C19CYP3A4CYP2D6
SCHEMBL601277 0.69 CYP3A4 (0.43) TLR7PTGS2PTGS1CYP2C19CYP3A4
SCHEMBL11274411 0.68 ESR1 (0.39) ESR1CYP2C19HSD17B10MEN1KMT2A
SCHEMBL603692 0.66 HSP90AA1 (0.44) TLR7CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL12764023 0.66 ESR1 (0.45) ESR1TSHRLMNAMEN1KMT2A
SCHEMBL31347570 0.66 NT5E (0.37) CYP2C19CYP3A4CYP2D6TSHRCRHBP
SCHEMBL26987221 0.66 NT5E (0.37) CYP2C19CYP3A4CYP2D6TSHRCRHBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798297-B1 Process for the preparation of 2-alkoxy-6-(trifluoromethyl)-pyrimidine-4-ol LONZA AG (CH) 2001-10-31 EP disclosed
US-5717096-A Process for the preparation of a 2-alkoxy-6-(trifluoromethyl)pyrimidin-4-ol LONZA AG (CH) 1998-02-10 US disclosed
EP-0798297-A1 Process for the preparation of 2-alkoxy-6-(triflourmethyl)-pyrimidin-4-ol LONZA AG (CH) 1997-10-01 EP disclosed