SCHEMBL7769575

SCHEMBL7769575

COC(=O)Oc1ccc2c(c1)OCC2(Cc1cc(C(C)(C)C)c(O)c(C(C)(C)C)c1)c1ccc2c(c1)C(C)(C)CCC2(C)C

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PPARG P37231 4/20 0.35
CYP26A1 O43174 8/20 0.34
CYP26B1 Q9NR63 6/20 0.34
CYP3A4 P08684 4/20 0.34
RXRA P19793 5/20 0.32
PTGS1 P23219 2/20 0.32
PTGS2 P35354 2/20 0.32
RXRB P28702 1/20 0.32
ALOX5 P09917 1/20 0.31
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7766320 0.91 CYP26B1 (0.37) PPARGCYP26A1CYP26B1CYP3A4RXRA
SCHEMBL6729485 0.87 CYP3A4 (0.41) CYP26A1CYP26B1CYP3A4RXRARXRB
SCHEMBL6736906 0.84 RXRA (0.45) CYP26A1CYP26B1RXRARXRBCNR2
SCHEMBL7770182 0.82 PPARG (0.37) PPARGCYP26A1CYP26B1CYP3A4RXRA
SCHEMBL7769865 0.80 RXRA (0.36) PPARGCYP26A1CYP26B1CYP3A4RXRA
SCHEMBL7770115 0.77 RXRA (0.38) PPARGCYP26A1CYP26B1CYP3A4RXRA
SCHEMBL7769613 0.77 RXRA (0.40) PPARGCYP26A1CYP26B1CYP3A4RXRA
SCHEMBL6730306 0.77 CYP3A4 (0.33) CYP26A1CYP3A4
SCHEMBL7773833 0.73 RXRA (0.39) PPARGCYP26A1CYP26B1CYP3A4RXRA
SCHEMBL7773881 0.73 CYP26B1 (0.42) PPARGCYP26A1CYP26B1CYP3A4RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0823903-B1 HETEROCYCLIC DIARYL COMPOUNDS, PHARMACEUTICAL AND COSMETIC COMPOSITIONS CONTAINING SAME, AND USES THEREOF CT INTERNAT DE RECH S (FR) 2001-07-18 EP claimed