SCHEMBL7770775

SCHEMBL7770775

COc1ccc(C(=O)N2CCC(C(SNC(=O)[C@@H](C)NC(=O)[C@@H]3CSCN3C(=O)OC(C)(C)C)C3CCCCC3)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.44
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
HSD17B10 Q99714 1/20 0.39
ABL1 P00519 1/20 0.39
RIN1 Q13671 1/20 0.39
ALDH1A1 P00352 2/20 0.38
GPR119 Q8TDV5 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TSHR P16473 1/20 0.37
UBE2M P61081 1/20 0.36
DCUN1D1 Q96GG9 1/20 0.36
ATM Q13315 1/20 0.36
STS P08842 1/20 0.36
MMP1 P03956 3/20 0.36
MMP3 P08254 3/20 0.36
MMP7 P09237 3/20 0.36
MMP9 P14780 3/20 0.36
MMP8 P22894 3/20 0.36
MMP13 P45452 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7772191 0.92 EPHX2 (0.41) EPHX2KMT2AMEN1HSD17B10ABL1
SCHEMBL7774527 0.88 MEN1 (0.43) KMT2AMEN1HSD17B10ALDH1A1SMN1; SMN2
SCHEMBL7105883 0.83 HSD17B10 (0.45) KMT2AMEN1HSD17B10GPR119TSHR
SCHEMBL7105591 0.82 MEN1 (0.43) KMT2AMEN1HSD17B10ALDH1A1ATM
SCHEMBL7110901 0.82 MEN1 (0.43) KMT2AMEN1HSD17B10ALDH1A1ATM
SCHEMBL7110470 0.82 MEN1 (0.43) KMT2AMEN1HSD17B10ALDH1A1ATM
SCHEMBL6705786 0.81 CYP2C19 (0.45) HSD17B10ALDH1A1GPR119SMN1; SMN2ATM
SCHEMBL5113474 0.79 CACNA1B (0.50) EPHX2KMT2AMEN1HSD17B10ABL1
SCHEMBL7105628 0.78 MEN1 (0.45) KMT2AMEN1HSD17B10ALDH1A1POLB
SCHEMBL5113479 0.77 EPHX2 (0.46) EPHX2KMT2AMEN1ABL1RIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1090912-A1 AMINO ACID DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2001-04-11 EP disclosed