SCHEMBL7773447

SCHEMBL7773447

CCOc1ccccc1N1CCN(CC(N)c2nc3ccc(F)cc3s2)CC1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 6/20 0.45
HTR1A P08908 3/20 0.45
SLC6A4 P31645 1/20 0.45
KCNH2 Q12809 1/20 0.45
DRD2 P14416 8/20 0.44
DRD4 P21917 6/20 0.44
DRD3 P35462 6/20 0.44
KDM4E B2RXH2 2/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
POLB P06746 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
HTR2C P28335 1/20 0.43
MAPT P10636 1/20 0.43
NLRP1 Q9C000 1/20 0.43
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL7848004 0.99 HTR7 (0.44) HTR7HTR1ASLC6A4KCNH2DRD2
SCHEMBL7856186 0.91 DRD3 (0.49) HTR1ADRD2DRD3KDM4EKMT2A
SCHEMBL7775362 0.89 ADRA1A (0.44) DRD4ADRA1DADRA1A
Bromide SCHEMBL7775341 0.88 ADRA1A (0.44) DRD4ADRA1DADRA1A
SCHEMBL27571993 0.87 NPC1 (0.38) HTR1ADRD2DRD3MAPTALDH1A1
SCHEMBL7776879 0.85 DRD2 (0.51) SLC6A4DRD2DRD3KMT2AMEN1
Bromide SCHEMBL7775396 0.85 DRD2 (0.50) SLC6A4DRD2DRD3KMT2AMEN1
SCHEMBL27577486 0.84 MAPT (0.42) KMT2AMEN1MAPTALDH1A1
Fumaric Acid SCHEMBL7855787 0.84 DRD3 (0.49) HTR7HTR1ADRD2DRD4DRD3
SCHEMBL27565726 0.82 NPC1 (0.44) HTR7SLC6A4KDM4EKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1117663-A2 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 2001-07-25 EP claimed
WO-2000018767-A2 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 2000-04-06 WO claimed
WO-2000018767-A9 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORP (US) 2001-04-19 WO disclosed