SCHEMBL7778629

SCHEMBL7778629

NCCNC(=O)COCC[O]

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
ALOX15 P16050 1/20 0.31
CYP2C19 P33261 1/20 0.31
HSD17B10 Q99714 1/20 0.31
KMT2A Q03164 2/20 0.31
CYP1A2 P05177 1/20 0.31
TSHR P16473 1/20 0.31
NFKB1 P19838 1/20 0.31
MAOB P27338 1/20 0.31
MEN1 O00255 1/20 0.30
BLM P54132 1/20 0.30
PMP22 Q01453 1/20 0.30
FAAH O00519 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7775664 0.89 PAOX (0.37) ALDH1A1KMT2ATSHRMEN1FAAH
SCHEMBL7778631 0.84 TSHR (0.35) ALDH1A1CYP2C9HPGDALOX15CYP2C19
SCHEMBL24040342 0.84 CA2 (0.34) ALDH1A1CYP2C9HPGDALOX15CYP2C19
SCHEMBL13018276 0.82 GLP1R (0.36) CYP2C19TSHR
SCHEMBL12730446 0.79 TSHR (0.42) ALDH1A1CYP2C9HPGDCYP2C19KMT2A
SCHEMBL12589997 0.79 TSHR (0.42) ALDH1A1CYP2C9HPGDCYP2C19KMT2A
SCHEMBL7771284 0.78 HSD17B10 (0.34) ALDH1A1HSD17B10KMT2ATSHRMEN1
SCHEMBL15765871 0.78 MEN1 (0.37) KMT2ATSHRMEN1
SCHEMBL14864751 0.78 NAMPT (0.42) ALDH1A1HPGDHSD17B10KMT2ATSHR
SCHEMBL14378850 0.78 POLB (0.38) ALDH1A1CYP2C9HPGDALOX15CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733045-B1 4,6-DIANILINO-PYRIMIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2001-08-16 EP disclosed
US-5880130-A TREATMENT OF CELL-PROLIFERATION DISEASES ZENECA LIMITED (GB) 1999-03-09 US disclosed
EP-0733045-A1 4,6-DIANILINO-PYRIMIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS TYROSINE KINASE INHIBITORS ZENECA LIMITED (GB) 1996-09-25 EP disclosed
WO-1995015952-A1 4,6-DIANILINO-PYRIMIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS TYROSINE KINASE INHIBITORS ZENECA LIMITED (GB) 1995-06-15 WO disclosed