SCHEMBL7779037

SCHEMBL7779037

C=C(C)C(=O)Nc1ccc(C(F)(F)F)cc1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.61
DHODH Q02127 1/20 0.59
TGM2 P21980 1/20 0.57
RXFP1 Q9HBX9 1/20 0.57
ALDH1A1 P00352 1/20 0.55
TRPV1 Q8NER1 2/20 0.54
RAB9A P51151 2/20 0.53
KIF11 P52732 1/20 0.53
NPC1 O15118 1/20 0.53
MEN1 O00255 2/20 0.53
HTT P42858 2/20 0.53
KMT2A Q03164 2/20 0.53
MAPT P10636 1/20 0.53
LMNA P02545 1/20 0.51
PTGS1 P23219 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12863513 0.87 RXFP1 (0.59) EPHX2DHODHTGM2RXFP1ALDH1A1
SCHEMBL3415035 0.85 EPHX2 (0.66) EPHX2DHODHTGM2ALDH1A1TRPV1
SCHEMBL2518624 0.85 EPHX2 (0.76) EPHX2DHODHTGM2ALDH1A1TRPV1
SCHEMBL439393 0.84 RXFP1 (0.74) RXFP1ALDH1A1RAB9ANPC1MEN1
SCHEMBL9078037 0.84 RXFP1 (0.59) EPHX2RXFP1ALDH1A1TRPV1RAB9A
SCHEMBL13274217 0.81 EPHX2 (0.59) EPHX2DHODHTGM2ALDH1A1TRPV1
SCHEMBL669442 0.81 EPHX2 (0.70) EPHX2DHODHTGM2ALDH1A1TRPV1
SCHEMBL10040308 0.81 DHODH (0.66) EPHX2DHODHTGM2ALDH1A1TRPV1
SCHEMBL8401862 0.81 DHODH (0.66) EPHX2DHODHTGM2ALDH1A1TRPV1
SCHEMBL7535310 0.80 TDP1 (0.62) RXFP1ALDH1A1RAB9AMEN1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107151224-A A kind of synthetic method of the alkyl-indol ketone derivatives of 3 methyl 3 江苏理工学院 2017-09-12 CN claimed
CN-107151224-A A kind of synthetic method of the alkyl-indol ketone derivatives of 3 methyl 3 江苏理工学院 2017-09-12 CN disclosed
CN-106831509-A A kind of synthetic method of Bicalutamide 西北师范大学 2017-06-13 CN disclosed
EP-1124795-A1 INHIBITORS OF THE EGF-RECEPTOR TYROSINE KINASE AND THEIR USE Parker Hughes Institute (US) 2001-08-22 EP disclosed
WO-2000056703-A1 INHIBITORS OF THE EGF-RECEPTOR TYROSINE KINASE AND THEIR USE PARKER HUGHES INSTITUTE (US) 2000-09-28 WO disclosed