SCHEMBL7779660

SCHEMBL7779660

C=CCc1ccc(-c2ccc(-c3ccc(C#N)cc3)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.47
HSD17B10 Q99714 1/20 0.47
LOXL2 Q9Y4K0 2/20 0.47
CYP2A6 P11509 1/20 0.47
MMP3 P08254 1/20 0.47
CYP3A4 P08684 2/20 0.43
CYP19A1 P11511 1/20 0.43
CYP1A2 P05177 1/20 0.43
POLB P06746 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
KIF11 P52732 3/20 0.42
ALDH1A1 P00352 1/20 0.42
TP53 P04637 1/20 0.42
ALOX15 P16050 1/20 0.42
ALOX12 P18054 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
IDO1 P14902 2/20 0.42
MMP12 P39900 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2352483 1.00 TSHR (0.47) TSHRHSD17B10LOXL2CYP2A6MMP3
SCHEMBL991288 0.94 LOXL2 (0.52) TSHRLOXL2CYP2A6CYP3A4CYP19A1
Bromide SCHEMBL28224574 0.92 LOXL2 (0.50) TSHRLOXL2CYP2A6CYP3A4CYP19A1
SCHEMBL20045130 0.88 LOXL2 (0.48) TSHRLOXL2CYP2A6CYP3A4CYP19A1
SCHEMBL11212791 0.86 CYP1A2 (0.39) TSHRHSD17B10LOXL2CYP2A6MMP3
Water SCHEMBL28100235 0.85 ALDH1A1 (0.54) TSHRHSD17B10CYP3A4CYP1A2POLB
SCHEMBL8927518 0.85 HRH3 (0.57) HRH3
SCHEMBL10586609 0.84 CYP11B1 (0.48) TSHRHSD17B10CYP3A4CYP19A1CYP1A2
SCHEMBL9063036 0.83 ALDH1A1 (0.52) TSHRLOXL2CYP2A6CYP3A4CYP19A1
SCHEMBL584333 0.82 ALDH1A1 (0.56) TSHRHSD17B10CYP3A4CYP1A2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE31715-E ESTERS OF 2-METHYLBUTYLPHENOL THE SECRETARY OF STATE FOR DEFENCE IN HER BRITANNIC MAJESTY'S GOVERNMENT OF THE UNITED KINGDOM OF GREAT BRITAIN AND NORTHERN IRELAND (GB) 1984-10-30 US claimed
US-4395350-A Liquid crystal mixtures HOFFMANN-LA ROCHE INC. (US) 1983-07-26 US claimed
US-4195916-A ELECTROOPTIC DISPLAY DEVICES, OPTICAL PHENOLIC ESTERS THE SECRETARY OF STATE FOR DEFENCE IN HER BRITANNIC MAJESTY'S GOVERNMENT OF THE UNITED KINGDOM OF GREAT BRITAIN AND NORTHERN IRELAND (GB) 1980-04-01 US claimed
JP-58034886-A None JP disclosed
EP-0851018-B1 Record display medium and use thereof DAINIPPON PRINTING CO LTD (JP) 2001-10-31 EP disclosed
EP-0790289-B1 Polymeric material for liquid crystal/polymer composite film, record display medium, and use thereof DAINIPPON PRINTING CO LTD (JP) 2001-09-05 EP disclosed
EP-0743350-B1 Smectic liquid crystal composition for recording display medium, recording display medium and use thereof DAINIPPON PRINTING CO LTD (JP) 2001-08-29 EP disclosed
US-6059993-A CONDUCTIVE SUBSTRATE; LIQUID CRYSTAL, COMPOSITE FILM DAI NIPPON PRINTING CO., LTD. (JP) 2000-05-09 US disclosed
US-5932137-A MIXTURE OF AROMATIC NITRILE AND AROMATIC ESTERS DAI NIPPON PRINTING CO., LTD. (JP) 1999-08-03 US disclosed
US-5851422-A Polymeric material for liquid crystal/polymer composite film, record display medium, and use thereof DAI NIPPON PRINTING CO., LTD. (JP) 1998-12-22 US disclosed
EP-0851018-A1 Record display medium and use thereof DAI NIPPON PRINTING CO., LTD. (JP) 1998-07-01 EP disclosed
US-4974941-A Process of aligning and realigning liquid crystal media HERCULES INCORPORATED (US) 1990-12-04 US disclosed
US-4583826-A Phenylethanes HOFFMANN-LA ROCHE INC. (US) 1986-04-22 US disclosed
EP-0058512-B1 LIQUID CRYSTAL COMPOUNDS EXHIBITING A SMALL DIELECTRIC ANISOTROPY AND LIQUID CRYSTAL MATERIALS AND DEVICES INCORPORATING SUCH COMPOUNDS The Secretary of State for Defence in Her Britannic Majesty's Government of the United Kingdom of Great Britain and (GB) 1986-01-15 EP disclosed
US-4556745-A BICYCOL(2.2.2) OCATANE RING THE SECRETARY OF STATE FOR DEFENCE IN HER BRITANNIC MAJESTY'S GOVERNMENT OF THE UNITED KINGDOM OF GREAT BRITAIN AND NORTHERN IRELAND (GB) 1985-12-03 US disclosed
US-4526704-A Esters containing phenylene and cyclohexylene rings HOFFMANN-LA ROCHE INC. (US) 1985-07-02 US disclosed
US-4395350-A Liquid crystal mixtures HOFFMANN-LA ROCHE INC. (US) 1983-07-26 US disclosed
JP-S5834886-A LIQUID CRYSTAL COMPOSITION SHARP CORP 1983-03-01 JP disclosed
EP-0058512-A1 Liquid crystal compounds exhibiting a small dielectric anisotropy and liquid crystal materials and devices incorporating such compounds The Secretary of State for Defence in Her Britannic Majesty's Government of the United Kingdom of Great Britain and (GB) 1982-08-25 EP disclosed
US-4149413-A THERMOCHROMIC THE SECRETARY OF STATE FOR DEFENCE IN HER BRITANNIC MAJESTY'S GOVERNMENT OF THE UNITED KINGDOM OF GREAT BRITAIN AND NORTHER IRELAND (GB) 1979-04-17 US disclosed