SCHEMBL7780580

SCHEMBL7780580

CC(NC(c1ccc(Cl)cc1)c1cccc(Nc2c(O)c(=O)c2=O)c1)c1cccc2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RCE1 Q9Y256 2/20 0.40
IDH1 O75874 1/20 0.38
THRA P10827 1/20 0.37
THRB P10828 1/20 0.37
S1PR3 Q99500 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ACKR3 P25106 1/20 0.36
PTGER4 P35408 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ACP3 P15309 1/20 0.35
ALOX5 P09917 3/20 0.35
PPARG P37231 3/20 0.35
CXCR2 P25025 1/20 0.34
GRIN2D O15399 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7785319 0.99 RCE1 (0.41) RCE1IDH1THRATHRBS1PR3
SCHEMBL7789338 0.93 RCE1 (0.45) RCE1LMNAALDH1A1GRIN2DGRIN3B
Hydrochloric Acid SCHEMBL7780764 0.92 RCE1 (0.47) RCE1MEN1KMT2AALDH1A1GRIN2D
SCHEMBL7787509 0.91 RCE1 (0.40) RCE1PTGER4ALDH1A1ALOX5PPARG
SCHEMBL7780400 0.91 RCE1 (0.40) RCE1PTGER4ALDH1A1ALOX5PPARG
Hydrochloric Acid SCHEMBL7785684 0.91 RCE1 (0.42) RCE1S1PR3PTGER4ALDH1A1CXCR2
Hydrochloric Acid SCHEMBL7787883 0.90 RCE1 (0.41) RCE1PTGER4ALDH1A1ALOX5PPARG
SCHEMBL7789329 0.89 MEN1 (0.40) RCE1THRATHRBMEN1KMT2A
SCHEMBL7789161 0.89 MEN1 (0.40) RCE1THRATHRBMEN1KMT2A
SCHEMBL7787711 0.87 CXCR2 (0.41) THRATHRBS1PR3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US claimed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP claimed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed