SCHEMBL7781846

SCHEMBL7781846

Cc1ccccc1C1OC=C(N2C(C(=O)OC(C)(C)C)=C(O)c3ccccc3S2(=O)=O)O1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.40
USP2 O75604 2/20 0.36
LMNA P02545 1/20 0.36
KDR P35968 1/20 0.36
ELANE P08246 2/20 0.32
PTGS1 P23219 3/20 0.32
PTGS2 P35354 3/20 0.32
ABCB11 O95342 1/20 0.32
GLA P06280 1/20 0.32
EDNRA P25101 1/20 0.32
KDM4E B2RXH2 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
ALOX15 P16050 1/20 0.32
NFKB1 P19838 1/20 0.32
CYP2C19 P33261 1/20 0.32
BLM P54132 1/20 0.32
SLC22A6 Q4U2R8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7787171 0.91 HSD11B1 (0.37) HSD11B1USP2LMNAKDRELANE
SCHEMBL6542004 0.72 HSD11B1 (0.45) HSD11B1USP2LMNAKDRELANE
SCHEMBL6542587 0.72 HSD11B1 (0.45) HSD11B1USP2LMNAELANEPTGS1
SCHEMBL6542415 0.72 EDNRA (0.42) HSD11B1USP2LMNAKDRPTGS1
SCHEMBL6542734 0.67 EDNRA (0.40) HSD11B1USP2LMNAKDREDNRA
SCHEMBL6542406 0.67 HSD11B1 (0.51) HSD11B1USP2LMNAKDRELANE
SCHEMBL7789463 0.65 CA9 (0.40) LMNAELANEKDM4ECYP2D6
SCHEMBL6542661 0.62 USP2 (0.47) HSD11B1USP2LMNAKDRPTGS1
SCHEMBL6541854 0.60 EDNRA (0.49) PTGS2EDNRAKDM4E
SCHEMBL6542493 0.59 LMNA (0.56) HSD11B1LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6252070-B1 REACTING ARYL BROMIDE WITH BUTYLLITHIUM AND ZINC BROMIDE TO GIVE ARYL ZINC BROMIDE; REACTING WITH CORRESPONDING BENZOTHIAZINE COMPOUND WARNER-LAMBERT COMPANY 2001-06-26 US disclosed