SCHEMBL7782959

SCHEMBL7782959

FC(F)(F)c1cccc(Cc2cc(Nc3cccc(C(F)(F)F)c3)ncn2)c1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.62
EGFR P00533 4/20 0.51
ERBB4 Q15303 1/20 0.51
AURKA O14965 2/20 0.49
GPR52 Q9Y2T5 5/20 0.48
KDM4E B2RXH2 1/20 0.48
ABCG2 Q9UNQ0 1/20 0.47
TNNI3K Q59H18 2/20 0.47
KDR P35968 2/20 0.47
BRAF P15056 1/20 0.47
MAPK14 Q16539 1/20 0.47
IDH2 P48735 1/20 0.47
SLC2A1 P11166 1/20 0.46
TSHR P16473 1/20 0.46
HTT P42858 1/20 0.46
MAPT P10636 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7781124 0.99 THRB (0.61) THRBEGFRERBB4AURKAGPR52
SCHEMBL7781150 0.88 THRB (0.55) THRBEGFRERBB4AURKAKDM4E
SCHEMBL7780162 0.87 GPR52 (0.48) THRBEGFRERBB4AURKAGPR52
Hydrochloric Acid SCHEMBL7776099 0.86 GPR52 (0.48) THRBEGFRERBB4AURKAGPR52
SCHEMBL7780190 0.86 THRB (0.47) THRBEGFRERBB4GPR52TNNI3K
Hydrochloric Acid SCHEMBL7783011 0.85 THRB (0.46) THRBEGFRERBB4GPR52TNNI3K
SCHEMBL30141460 0.84 THRB (0.65) THRBEGFRERBB4AURKAGPR52
SCHEMBL1387447 0.83 THRB (0.80) THRBEGFRERBB4AURKAKDM4E
SCHEMBL374332 0.80 THRB (0.74) THRBEGFRERBB4AURKAKDM4E
SCHEMBL7776064 0.78 HTR2B (0.46) GPR52MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0972770-B1 Acaricidal and insecticidal substituted pyrimidines and a process for the preparation thereof BASF AG (DE) 2001-09-19 EP claimed
US-6281219-B1 4,6-BIS-ARYL-PYRIMIDINES WHEREIN THE AROMATIC GROUPS ARE ATTACHED VIA TWO LINKING GROUPS WHICH ARE DIFFERENT FROM ONE ANOTHER. AMERICAN CYANAMID CO. 2001-08-28 US claimed
EP-0972770-A1 Acaricidal and insecticidal substituted pyrimidines and a process for the preparation thereof American Cyanamid Company (US) 2000-01-19 EP claimed