SCHEMBL7781150

SCHEMBL7781150

FC(F)(F)c1cccc(Nc2cc(Cc3ccc(Cl)c(Cl)c3)ncn2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.55
EGFR P00533 5/20 0.46
ERBB4 Q15303 1/20 0.46
AURKA O14965 2/20 0.44
MAPT P10636 2/20 0.44
ALDH1A1 P00352 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
P2RX3 P56373 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ABCG2 Q9UNQ0 1/20 0.42
CTSC P53634 3/20 0.42
TNNI3K Q59H18 2/20 0.42
TRPV1 Q8NER1 1/20 0.41
IDH2 P48735 1/20 0.41
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
BRAF P15056 1/20 0.41
KDR P35968 1/20 0.41
MAPK14 Q16539 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7782959 0.88 THRB (0.62) THRBEGFRERBB4AURKAMAPT
Hydrochloric Acid SCHEMBL7781124 0.87 THRB (0.61) THRBEGFRERBB4AURKAKDM4E
SCHEMBL7780190 0.85 THRB (0.47) THRBEGFRERBB4TNNI3KTRPV1
SCHEMBL7780172 0.84 KMO (0.43) ALDH1A1BRAFKDR
Hydrochloric Acid SCHEMBL7783011 0.84 THRB (0.46) THRBEGFRERBB4TNNI3KTRPV1
SCHEMBL7781111 0.81 STK17B (0.41) CTSCBRAFKDR
Hydrochloric Acid SCHEMBL7783014 0.81 STK17B (0.40) CTSCBRAFKDR
SCHEMBL30141460 0.78 THRB (0.65) THRBEGFRERBB4AURKAKDM4E
SCHEMBL1387447 0.78 THRB (0.80) THRBEGFRERBB4AURKAKDM4E
SCHEMBL7780162 0.77 GPR52 (0.48) THRBEGFRERBB4AURKAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0972770-B1 Acaricidal and insecticidal substituted pyrimidines and a process for the preparation thereof BASF AG (DE) 2001-09-19 EP claimed
US-6281219-B1 4,6-BIS-ARYL-PYRIMIDINES WHEREIN THE AROMATIC GROUPS ARE ATTACHED VIA TWO LINKING GROUPS WHICH ARE DIFFERENT FROM ONE ANOTHER. AMERICAN CYANAMID CO. 2001-08-28 US claimed
EP-0972770-A1 Acaricidal and insecticidal substituted pyrimidines and a process for the preparation thereof American Cyanamid Company (US) 2000-01-19 EP claimed
EP-0972770-B1 Acaricidal and insecticidal substituted pyrimidines and a process for the preparation thereof BASF AG (DE) 2001-09-19 EP disclosed
US-6281219-B1 4,6-BIS-ARYL-PYRIMIDINES WHEREIN THE AROMATIC GROUPS ARE ATTACHED VIA TWO LINKING GROUPS WHICH ARE DIFFERENT FROM ONE ANOTHER. AMERICAN CYANAMID CO. 2001-08-28 US disclosed
EP-0972770-A1 Acaricidal and insecticidal substituted pyrimidines and a process for the preparation thereof American Cyanamid Company (US) 2000-01-19 EP disclosed