SCHEMBL7784559

SCHEMBL7784559

N#Cc1ccc([N]CCc2ccccc2Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 1/20 0.49
HTR3B O95264 1/20 0.49
HTR3A P46098 1/20 0.49
HTR3D Q70Z44 1/20 0.49
HTR3C Q8WXA8 1/20 0.49
TAAR1 Q96RJ0 3/20 0.41
AOC3 Q16853 1/20 0.39
HSD11B1 P28845 2/20 0.37
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
KCNH2 Q12809 1/20 0.36
TSHR P16473 1/20 0.35
PNMT P11086 1/20 0.35
IDO1 P14902 1/20 0.35
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
PYCR1 P32322 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7784561 0.72 TAAR1 (0.49) TAAR1AOC3
SCHEMBL15445886 0.71 SLC5A2 (0.46) HSD11B1SLC6A2SLC6A4SLC6A3TSHR
SCHEMBL17217371 0.68 KMT2A (0.42) HSD11B1SLC6A4IDO1MAOAMAOB
SCHEMBL17217374 0.68 KMT2A (0.42) HSD11B1SLC6A4IDO1MAOAMAOB
SCHEMBL11114725 0.67 TAAR1 (0.50) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL1343862 0.66 TAAR1 (0.54) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL6740216 0.66 TAAR1 (0.71) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL6961980 0.66 MIF (0.55) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL5480950 0.66 HTR3E (0.53) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8176728 0.66 TSHR (0.46) TSHRNOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150963-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM Aventis Pharma Deutschland GmbH (DE) 2001-11-07 EP disclosed
WO-2000046214-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-08-10 WO disclosed