SCHEMBL7784720

SCHEMBL7784720

CC(NC(c1ccc(Cl)cc1)c1cccc([N+](=O)[O-])c1)c1cc(F)cc(F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
MEN1 O00255 5/20 0.39
KMT2A Q03164 5/20 0.39
HPGD P15428 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
MGAM O43451 1/20 0.37
CNR1 P21554 1/20 0.37
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7785724 1.00 ALDH1A1 (0.40) ALDH1A1TDP1CYP3A4CYP2D6SLC6A2
SCHEMBL7789050 0.93 ALDH1A1 (0.40) ALDH1A1TDP1CYP3A4CYP2D6SLC6A2
SCHEMBL27533527 0.92 MEN1 (0.40) ALDH1A1CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL7787532 0.92 MEN1 (0.40) ALDH1A1CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL7785105 0.91 CRHBP (0.44) ALDH1A1MEN1KMT2AHPGDL3MBTL1
SCHEMBL7785576 0.91 CRHBP (0.44) ALDH1A1MEN1KMT2AHPGDL3MBTL1
SCHEMBL7787830 0.90 AKR1C3 (0.41) ALDH1A1TDP1CYP3A4CYP2D6SLC6A2
SCHEMBL7785645 0.90 AKR1C3 (0.41) ALDH1A1TDP1CYP3A4CYP2D6SLC6A2
SCHEMBL7780592 0.90 HTT (0.46) ALDH1A1CYP3A4MEN1KMT2AHPGD
SCHEMBL27540162 0.90 HTT (0.46) ALDH1A1CYP3A4MEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
CN-1287117-A Cyclobutene derivatives, preparation method and therapeutic use thereof SANKYO CO (JP) 2001-03-14 CN disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed