SCHEMBL7784867

SCHEMBL7784867

COC(=O)c1ccc2[nH]cc(CCCCN3CCN(c4cc(=O)oc5cc(OC)ccc45)CC3)c2c1

nearest known ligand 0.70

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.59
ADRA2B P18089 2/20 0.59
ADRA2C P18825 2/20 0.59
ADRA1D P25100 2/20 0.59
ADRA1A P35348 2/20 0.59
ADRA1B P35368 2/20 0.59
HTR1A P08908 3/20 0.54
DRD2 P14416 1/20 0.54
HTR2A P28223 1/20 0.54
SLC6A4 P31645 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7785348 0.95 ADRA2A (0.52) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL5204281 0.93 ADRA2A (0.60) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL7784871 0.92 SLC6A4 (0.53) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL7785392 0.91 SLC6A4 (0.53) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL7780259 0.91 SLC6A4 (0.53) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL5201347 0.90 ADRA2A (0.59) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL7787588 0.90 SLC6A4 (0.56) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL7788884 0.89 HTR1A (0.54) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL5204284 0.89 ADRA2A (0.59) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL7784858 0.88 ADRA2A (0.53) ADRA2AADRA2BADRA2CADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251908-B1 Piperazine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 2001-06-26 US disclosed