SCHEMBL7784876

SCHEMBL7784876

Cc1cc2oc(=O)ccc2cc1N1CCN(CCCCc2c[nH]c3cc(C(=O)O)ccc23)CC1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.43
ADRA2A P08913 2/20 0.42
ADRA2B P18089 2/20 0.42
ADRA2C P18825 2/20 0.42
ADRA1D P25100 2/20 0.42
ADRA1A P35348 2/20 0.42
ADRA1B P35368 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5203742 0.94 ADRA2A (0.49) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL7784879 0.92 SLC6A4 (0.49) HTR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL7780289 0.91 HTR1A (0.45) HTR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL7780297 0.91 ADRA2A (0.46) HTR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL7780314 0.91 ADRA2A (0.43) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL7788865 0.90 HTR1A (0.45) HTR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL8124382 0.87 HTR1A (0.45) HTR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL7785338 0.86 HTR1A (0.56) HTR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL7787566 0.85 SLC6A4 (0.56) HTR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL7788881 0.85 HTR1A (0.51) HTR1AADRA2AADRA2BADRA2CADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1093127-C Piperazine derivatives MERCK PATENT GMBH (DE) 2002-10-23 CN disclosed
US-6251908-B1 Piperazine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 2001-06-26 US disclosed
CN-1264379-A Piperazine derivatives MERCK PATENT GMBH (DE) 2000-08-23 CN disclosed