SCHEMBL7784955

SCHEMBL7784955

O=C(O)C1(C(=O)c2ccccc2)CCNCC1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.44
OPRM1 P35372 2/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 3/20 0.40
ALDH1A1 P00352 2/20 0.40
USP2 O75604 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP2D6 P10635 2/20 0.39
CYP1A2 P05177 1/20 0.39
DPP9 Q86TI2 1/20 0.38
DPP7 Q9UHL4 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
HDAC1 Q13547 1/20 0.38
DAO P14920 1/20 0.37
NAPRT Q6XQN6 1/20 0.37
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7840180 0.81 GABRD (0.53) LMNA
SCHEMBL5558534 0.81 AKR1C1 (0.47) LMNATSHRALDH1A1CYP2D6DAO
SCHEMBL27963066 0.79 SIGMAR1 (0.46) SIGMAR1OPRM1LMNATSHRALDH1A1
SCHEMBL11761384 0.79 OPRM1 (0.48) SIGMAR1OPRM1LMNATSHRALDH1A1
SCHEMBL20228048 0.78 SIGMAR1 (0.44) SIGMAR1OPRM1LMNATSHRALDH1A1
SCHEMBL18321798 0.78 SIGMAR1 (0.44) SIGMAR1OPRM1LMNATSHRALDH1A1
SCHEMBL7312326 0.76 OPRM1 (0.56) SIGMAR1OPRM1HDAC1
SCHEMBL825722 0.75 KDM4E (0.38) OPRM1TSHRCYP2D6CYP1A2
SCHEMBL23467203 0.74 SLC6A2 (0.47) SIGMAR1OPRM1LMNACYP2D6SLC6A2
SCHEMBL14637529 0.74 OPRM1 (0.43) SIGMAR1OPRM1LMNATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140838-A1 1, 4-PIPERAZINE DERIVATIVES HAVING 5HT1A RECEPTOR ACTIVITY AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-10 EP disclosed
WO-2000035878-A1 1,4-PIPERAZINE DERIVATIVES HAVING 5HT1A RECEPTOR ACTIVITY AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-22 WO disclosed