SCHEMBL7785166

SCHEMBL7785166

CON=C(C(=O)N(C)C)C(C)=NN(C)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 8/20 0.34
KMT2A Q03164 8/20 0.34
MAPT P10636 6/20 0.34
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
TDP1 Q9NUW8 2/20 0.34
LMNA P02545 2/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ALOX12 P18054 1/20 0.32
TSHR P16473 1/20 0.32
MTNR1A P48039 1/20 0.31
MTNR1B P49286 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7785163 1.00 MEN1 (0.34) MEN1KMT2AMAPTNPC1RAB9A
SCHEMBL8537305 0.75 RAB9A (0.43) MEN1KMT2AMAPTNPC1RAB9A
SCHEMBL7785156 0.73 ALDH1A1 (0.41) MAPTNPC1RAB9ASMN1; SMN2L3MBTL1
SCHEMBL7785155 0.73 ALDH1A1 (0.41) MAPTNPC1RAB9ASMN1; SMN2L3MBTL1
SCHEMBL7787058 0.71 THRB (0.36) MAPTSMN1; SMN2TDP1TSHR
SCHEMBL7787055 0.71 THRB (0.36) MAPTSMN1; SMN2TDP1TSHR
SCHEMBL7787357 0.69
SCHEMBL7787356 0.69
SCHEMBL11509828 0.67
SCHEMBL8537307 0.67 TSHR (0.42) KMT2AMAPTNPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251949-B1 AGRICULTURAL FUNGICIDE, ALSO HAS TACHYKININ RECEPTOR ANTAGONSITIC EFFECT, AND THUS IS USEFUL AS PHARMECEUTICAL SHIONOGI & CO., LTD. (JP) 2001-06-26 US disclosed
US-6096741-A FUNGICIDES, TACHYKININ ANTAGONIST SHIONOGI & CO., LTD. (JP) 2000-08-01 US disclosed
EP-0940388-A1 OXIME DERIVATIVES, HYDRAZONE DERIVATIVES, AND USE THEREOF SHIONOGI & CO., LTD. (JP) 1999-09-08 EP disclosed