SCHEMBL7785246

SCHEMBL7785246

CON=C(C)c1ccc(Br)cc1F.CON=CC(=NOC)c1ccc(F)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.34
MAPT P10636 2/20 0.32
KDM4E B2RXH2 1/20 0.32
DGAT1 O75907 1/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TRPA1 O75762 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7575127 0.89 SLC6A4 (0.39) SLC6A4MAPTKDM4EDGAT1NPC1
SCHEMBL6819500 0.79 DGAT1 (0.47) SLC6A4MAPTKDM4EDGAT1NPC1
SCHEMBL6819503 0.79 DGAT1 (0.47) SLC6A4MAPTKDM4EDGAT1NPC1
SCHEMBL7872121 0.77 CES2 (0.42) MAPTKDM4EALDH1A1RAB9ASMN1; SMN2
SCHEMBL6811082 0.77 MAPT (0.45) MAPTNPC1GAARAB9AKMT2A
SCHEMBL6811077 0.77 MAPT (0.45) MAPTNPC1GAARAB9AKMT2A
SCHEMBL6814924 0.74 CES2 (0.47) MAPTKDM4EALDH1A1LMNARAB9A
SCHEMBL6814922 0.74 CES2 (0.47) MAPTKDM4EALDH1A1LMNARAB9A
SCHEMBL7862677 0.70 SLC6A4 (0.36) SLC6A4DGAT1NPC1ALDH1A1LMNA
SCHEMBL7862674 0.70 RAB9A (0.46) SLC6A4MAPTDGAT1NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144397-A3 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING PHENYLENEDIAMINE GROUP Wyeth (US) 2002-09-11 EP disclosed
EP-1144397-A2 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-17 EP disclosed
WO-2000034258-A2 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-15 WO disclosed