SCHEMBL7785330

SCHEMBL7785330

O=S(=O)(Oc1ccc(-c2ccc(OS(=O)(=O)C(F)(F)F)c(Br)c2)cc1Br)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 13/20 0.39
PTGS2 P35354 3/20 0.36
PTGS1 P23219 2/20 0.36
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
DRD2 P14416 1/20 0.34
DRD1 P21728 1/20 0.34
DRD4 P21917 1/20 0.34
DRD5 P21918 1/20 0.34
DRD3 P35462 1/20 0.34
PIM1 P11309 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8502379 0.83 EPAS1 (0.47) EPAS1CA1CA2
SCHEMBL20193401 0.83 EPAS1 (0.37) EPAS1CA1CA2DRD2DRD1
SCHEMBL29134970 0.81 EPAS1 (0.43) EPAS1CA1CA2
SCHEMBL18183948 0.81 EPAS1 (0.36) EPAS1CA1CA2DRD2DRD1
SCHEMBL5787332 0.80 ALDH1A1 (0.43) EPAS1PTGS2PTGS1CA1CA2
SCHEMBL2860586 0.78 CA1 (0.42) EPAS1CA1CA2DRD2DRD1
SCHEMBL31265243 0.78 CA1 (0.42) EPAS1CA1CA2DRD2DRD1
SCHEMBL12275709 0.78 CA2 (0.37) EPAS1CA1CA2DRD2DRD1
SCHEMBL12294158 0.78 CA2 (0.37) EPAS1CA1CA2DRD2DRD1
SCHEMBL2469383 0.76 NOTUM (0.57) CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0854849-B1 ETHYNYL SUBSTITUTED AROMATIC COMPOUNDS, SYNTHESIS, POLYMERS AND USES THEREOF DOW CHEMICAL CO (US) 2001-10-31 EP disclosed
US-6252001-B1 ACETYLENIC POLYMER THE DOW CHEMICAL COMPANY 2001-06-26 US disclosed
US-6121495-A Ethynyl substituted aromatic compounds, synthesis, polymers and uses thereof THE DOW CHEMICAL COMPANY (US) 2000-09-19 US disclosed