SCHEMBL7785667

SCHEMBL7785667

CON=CC(=NOC)c1ccc(F)c(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.38
TAS1R1 Q7RTX1 2/20 0.38
TAS1R2 Q8TE23 2/20 0.38
PTPN7 P35236 6/20 0.37
DUSP3 P51452 6/20 0.37
HDAC8 Q9BY41 1/20 0.34
KCNQ3 O43525 1/20 0.33
KCNQ2 O43526 1/20 0.33
KCNE1 P15382 1/20 0.33
KCNQ1 P51787 1/20 0.33
KIF11 P52732 1/20 0.32
NOTUM Q6P988 1/20 0.32
PPARD Q03181 1/20 0.32
PPARA Q07869 1/20 0.32
VNN1 O95497 3/20 0.32
P4HB P07237 1/20 0.31
IDO1 P14902 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6814822 0.78 NPFFR2 (0.42) TAS1R3TAS1R1TAS1R2PTPN7DUSP3
SCHEMBL6814827 0.78 NPFFR2 (0.42) TAS1R3TAS1R1TAS1R2PTPN7DUSP3
SCHEMBL7784450 0.76 PDE2A (0.38) IDO1
SCHEMBL27472637 0.74 PTPN7 (0.39) TAS1R3TAS1R1TAS1R2PTPN7DUSP3
SCHEMBL7784407 0.73 NOTUM (0.33) NOTUMVNN1
SCHEMBL7872121 0.69 CES2 (0.42)
SCHEMBL14012580 0.68 NOTUM (0.64) TAS1R3TAS1R1TAS1R2HDAC8KCNQ3
SCHEMBL22561756 0.68 NOTUM (0.47) TAS1R3TAS1R1TAS1R2PTPN7DUSP3
SCHEMBL752590 0.68 NOTUM (0.64) TAS1R3TAS1R1TAS1R2HDAC8KCNQ3
SCHEMBL7847467 0.68 GAA (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1137647-A1 THIOUREA INHIBITORS OF HERPES VIRUSES AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-04 EP disclosed
EP-1137633-A2 ACETAMIDE AND SUBSTITUTED ACETAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-04 EP disclosed
US-6255349-B1 PREVENTION REPRODUCTION; VIRICIDES AMERICAN HOME PRODUCTS CORPORATION 2001-07-03 US disclosed
WO-2000034268-A1 THIOUREA INHIBITORS OF HERPES VIRUSES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-15 WO disclosed
WO-2000034237-A2 ACETAMIDE AND SUBSTITUTED ACETAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-15 WO disclosed