SCHEMBL7786980

SCHEMBL7786980

O=C(NCc1ccc(C(=O)N[C@H](CO)Cc2ccccc2)cc1)c1ccc2ccccc2c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.65
HDAC3 O15379 2/20 0.64
HDAC1 Q13547 2/20 0.64
HDAC2 Q92769 2/20 0.64
HDAC4 P56524 1/20 0.64
HDAC7 Q8WUI4 1/20 0.64
HDAC10 Q969S8 1/20 0.64
HDAC11 Q96DB2 1/20 0.64
HDAC8 Q9BY41 1/20 0.64
HDAC6 Q9UBN7 1/20 0.64
HDAC9 Q9UKV0 1/20 0.64
HDAC5 Q9UQL6 1/20 0.64
PIN1 Q13526 8/20 0.60
ROCK2 O75116 1/20 0.56
RPS6KA5 O75582 1/20 0.56
RPS6KA4 O75676 1/20 0.56
PRKACA P17612 1/20 0.56
MAPK1 P28482 1/20 0.56
GSK3A P49840 1/20 0.56
GSK3B P49841 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7789870 0.86 PIN1 (0.60) NR1H4PIN1ROCK2RPS6KA5RPS6KA4
SCHEMBL7789871 0.86 PIN1 (0.60) NR1H4PIN1ROCK2RPS6KA5RPS6KA4
SCHEMBL7789993 0.84 NR1H4 (0.62) NR1H4HDAC3HDAC1HDAC2HDAC4
SCHEMBL14894197 0.83 NR1H4 (0.85) NR1H4HDAC3HDAC1HDAC2HDAC4
SCHEMBL7787818 0.83 OPRK1 (0.61) HDAC2HDAC8HDAC6PIN1ROCK2
SCHEMBL7787816 0.83 OPRK1 (0.61) HDAC2HDAC8HDAC6PIN1ROCK2
SCHEMBL6943275 0.82 NR1H4 (0.60) NR1H4HDAC3HDAC1HDAC2HDAC4
SCHEMBL7782138 0.82 NPC1 (0.59) NR1H4PIN1ROCK2RPS6KA5RPS6KA4
SCHEMBL7789811 0.82 PIN1 (0.55) PIN1ROCK2RPS6KA5RPS6KA4PRKACA
SCHEMBL7789810 0.82 PIN1 (0.55) PIN1ROCK2RPS6KA5RPS6KA4PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed