SCHEMBL7789870

SCHEMBL7789870

O=C(Nc1ccc(C(=O)N[C@H](CO)Cc2ccccc2)cc1)c1ccc2ccccc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 9/20 0.60
NR1H4 Q96RI1 2/20 0.59
ROCK2 O75116 1/20 0.56
RPS6KA5 O75582 1/20 0.56
RPS6KA4 O75676 1/20 0.56
PRKACA P17612 1/20 0.56
MAPK1 P28482 1/20 0.56
GSK3A P49840 1/20 0.56
GSK3B P49841 1/20 0.56
IRAK1 P51617 1/20 0.56
PRKX P51817 1/20 0.56
ROCK1 Q13464 1/20 0.56
PRKG1 Q13976 1/20 0.56
PKN2 Q16513 1/20 0.56
CLK4 Q9HAZ1 1/20 0.56
SGK2 Q9HBY8 1/20 0.56
DEGS1 O15121 1/20 0.55
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
NPC1 O15118 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7789871 1.00 PIN1 (0.60) PIN1NR1H4ROCK2RPS6KA5RPS6KA4
SCHEMBL7782138 0.91 NPC1 (0.59) PIN1NR1H4ROCK2RPS6KA5RPS6KA4
SCHEMBL6946318 0.90 PIN1 (0.66) PIN1NR1H4DEGS1MEN1KMT2A
SCHEMBL7786980 0.86 NR1H4 (0.65) PIN1NR1H4ROCK2RPS6KA5RPS6KA4
SCHEMBL6802171 0.84 DEGS1 (0.57) PIN1ROCK2RPS6KA5RPS6KA4PRKACA
SCHEMBL6802167 0.84 DEGS1 (0.57) PIN1ROCK2RPS6KA5RPS6KA4PRKACA
SCHEMBL6945342 0.83 PIN1 (0.55) PIN1NR1H4DEGS1MEN1KMT2A
SCHEMBL7789992 0.83 NR1H4 (0.58) PIN1NR1H4DEGS1MEN1KMT2A
SCHEMBL7789989 0.83 NR1H4 (0.58) PIN1NR1H4DEGS1MEN1KMT2A
SCHEMBL7789327 0.81 ALDH1A1 (0.57) PIN1ROCK2RPS6KA5RPS6KA4PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed