SCHEMBL7789425

SCHEMBL7789425

COc1ccc(C(Br)c2cccc([N+](=O)[O-])c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 1/20 0.55
MAPT P10636 4/20 0.52
ALDH1A1 P00352 2/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
MAPK1 P28482 2/20 0.50
NPSR1 Q6W5P4 1/20 0.50
TDP1 Q9NUW8 1/20 0.49
SMN1; SMN2 Q16637 4/20 0.48
LMNA P02545 3/20 0.48
ACP3 P15309 1/20 0.46
TP53 P04637 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
PKM P14618 1/20 0.45
POLB P06746 1/20 0.45
HTT P42858 1/20 0.45
APP P05067 1/20 0.44
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11442189 0.85 APP (0.55) MAPTALDH1A1NPC1RAB9AMAPK1
SCHEMBL11432821 0.84 TSHR (0.61) MAPTALDH1A1TDP1SMN1; SMN2LMNA
SCHEMBL7785663 0.83 NFE2L2 (0.55) NFE2L2MAPTALDH1A1NPC1RAB9A
SCHEMBL7801278 0.83 NFE2L2 (0.55) NFE2L2MAPTALDH1A1NPC1RAB9A
Hydrochloric Acid SCHEMBL7787525 0.82 NFE2L2 (0.53) NFE2L2MAPTALDH1A1NPC1RAB9A
Trimethylammonium SCHEMBL28709705 0.81 NFE2L2 (0.52) NFE2L2MAPTALDH1A1NPC1RAB9A
SCHEMBL8402461 0.78 NFE2L2 (0.47) NFE2L2MAPTALDH1A1NPC1RAB9A
SCHEMBL7788967 0.78 MAPK1 (0.51) NFE2L2MAPTALDH1A1NPC1RAB9A
SCHEMBL5243706 0.77 TSHR (0.52) NFE2L2MAPTALDH1A1TDP1SMN1; SMN2
SCHEMBL15325817 0.77 ALDH1A1 (0.58) NFE2L2MAPTALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
CN-1287117-A Cyclobutene derivatives, preparation method and therapeutic use thereof SANKYO CO (JP) 2001-03-14 CN disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed