SCHEMBL7790904

SCHEMBL7790904

C#CCn1nc(-c2ccc(SC)cc2)c(-c2ccc(F)cc2)c1C(F)(F)F.CSc1ccc(-c2n[nH]c(C(F)(F)F)c2-c2ccc(F)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.43
PTGS1 P23219 1/20 0.43
GYS1 P13807 5/20 0.39
MAPK13 O15264 4/20 0.33
MAPK12 P53778 4/20 0.33
MAPK11 Q15759 4/20 0.33
MAPK14 Q16539 4/20 0.33
GCGR P47871 3/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
LCK P06239 1/20 0.33
RET P07949 1/20 0.33
ALOX5 P09917 1/20 0.33
PRKACA P17612 1/20 0.33
RPS6KB1 P23443 1/20 0.33
MATK P42679 1/20 0.33
FRK P42685 1/20 0.33
MAPK9 P45984 1/20 0.33
CSNK1A1 P48729 1/20 0.33
CSNK1D P48730 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7780920 0.90 PTGS2 (0.51) PTGS2PTGS1MAPK13MAPK12MAPK11
SCHEMBL7777792 0.82 GYS1 (0.54) PTGS2PTGS1GYS1MAPK13MAPK12
SCHEMBL7773294 0.78 PTGS2 (0.60) PTGS2PTGS1
SCHEMBL7778238 0.77 PTGS2 (0.60) PTGS2PTGS1MAPK14ALOX5GABRP
SCHEMBL7773251 0.74 PTGS2 (0.76) PTGS2PTGS1
SCHEMBL7773122 0.72 PTGS2 (0.74) PTGS2PTGS1
SCHEMBL7777945 0.72 MAPK14 (0.38) PTGS2PTGS1MAPK13MAPK12MAPK11
SCHEMBL7777683 0.72 MAPK14 (0.49) PTGS2PTGS1MAPK13MAPK12MAPK11
SCHEMBL8953773 0.71 GYS1 (0.54) PTGS2PTGS1GYS1MAPK14GCGR
SCHEMBL8758606 0.69 GYS1 (0.38) PTGS2PTGS1GYS1MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0772597-B1 3,4-SUBSTITUTED PYRAZOLES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2001-12-12 EP disclosed