SCHEMBL7791989

SCHEMBL7791989

CCOc1ccc2c(c1)C(=O)c1cccc(OCCCN3CCCC3)c1-2

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
TSHR P16473 1/20 0.53
HRH3 Q9Y5N1 8/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
KDM4E B2RXH2 2/20 0.49
HTT P42858 1/20 0.49
ADORA2A P29274 5/20 0.48
ADORA2B P29275 4/20 0.48
ADORA1 P30542 4/20 0.48
ADORA3 P0DMS8 3/20 0.48
KCNH2 Q12809 1/20 0.48
DRD2 P14416 1/20 0.46
DRD3 P35462 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27514547 0.97 ALDH1A1 (0.53) ALDH1A1TSHRHRH3L3MBTL1KDM4E
SCHEMBL7796470 0.95 KDM4E (0.50) ALDH1A1TSHRHRH3KDM4EHTT
SCHEMBL7796403 0.94 HRH3 (0.53) ALDH1A1TSHRHRH3L3MBTL1KDM4E
SCHEMBL7795710 0.94 HRH3 (0.51) ALDH1A1TSHRHRH3KDM4EHTT
SCHEMBL7794709 0.93 HRH3 (0.55) ALDH1A1TSHRHRH3L3MBTL1KDM4E
SCHEMBL7792408 0.93 HRH3 (0.52) ALDH1A1TSHRHRH3L3MBTL1KDM4E
SCHEMBL27514549 0.91 HRH3 (0.50) HRH3ADORA2AADORA2BADORA1ADORA3
SCHEMBL27494797 0.91 HRH3 (0.53) HRH3L3MBTL1KDM4EADORA2AADORA2B
SCHEMBL7792385 0.90 HRH3 (0.55) ALDH1A1HRH3KDM4EKCNH2
SCHEMBL7786144 0.89 LTA4H (0.51) ALDH1A1HRH3L3MBTL1KDM4EADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906268-B1 ALKYLOXYAMINO SUBSTITUTED FLUORENONES AND THEIR USE AS PROTEIN KINASE C INHIBITORS AVENTIS PHARMA INC (US) 2001-11-28 EP disclosed
US-6004959-A HYPOTENSIVE, ANTITUMOR, ANTIINFLAMMATORY AND ANTIASTHMATIC AGENTS; ANGIOGENESIS AND ALVEOLAR MACROPHAGE ACTIVATION INHIBITORS HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US disclosed