SCHEMBL7792264

SCHEMBL7792264

COc1ccc(CN)cc1.O=Cc1ccc(Oc2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
CYP2A6 P11509 1/20 0.56
LTA4H P09960 2/20 0.53
RAB9A P51151 3/20 0.52
KDM4E B2RXH2 1/20 0.52
HTT P42858 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
NPC1 O15118 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
TTR P02766 1/20 0.49
MAOB P27338 3/20 0.46
ST14 Q9Y5Y6 1/20 0.46
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
TRPA1 O75762 1/20 0.45
PARP10 Q53GL7 1/20 0.43
PARP3 Q9Y6F1 1/20 0.43
SRD5A2 P31213 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzaldehyde SCHEMBL7792134 0.91 ALDH1A1 (0.58) ALDH1A1CYP2A6LTA4HRAB9AKDM4E
SCHEMBL7792799 0.90 MAOB (0.52) ALDH1A1CYP2A6LTA4HRAB9AKDM4E
SCHEMBL7798169 0.90 NPC1 (0.63) ALDH1A1CYP2A6LTA4HRAB9AKDM4E
SCHEMBL7792654 0.89 TAAR1 (0.58) ALDH1A1CYP2A6LTA4HRAB9AKDM4E
Anisaldehyde SCHEMBL6814373 0.82 ALDH1A1 (0.83) ALDH1A1CYP2A6LTA4HRAB9ANPC1
SCHEMBL7792570 0.81 NPC1 (0.59) ALDH1A1LTA4HRAB9AKDM4EHTT
SCHEMBL7792557 0.81 MAOB (0.52) ALDH1A1RAB9AKDM4EHTTSMN1; SMN2
SCHEMBL920324 0.80 ST14 (0.68) ALDH1A1LTA4HKDM4EHTTSMN1; SMN2
SCHEMBL527049 0.80 ALDH1A1 (0.86) ALDH1A1CYP2A6LTA4HKDM4ESMN1; SMN2
Benzaldehyde SCHEMBL7798573 0.79 TAAR1 (0.66) ALDH1A1CYP2A6LTA4HRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1076649-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 2001-02-21 EP disclosed
US-6127381-A A MELANOCORTIN RECEPTOR LIGAND FOR REGULATING FOOD INTAKE AND BODY WEIGHT, REGULATING CYTOKINE ACTIVITY, ANTI-INFLAMMATORY ACTIVITY LION BIOSCIENCE AG (DE) 2000-10-03 US disclosed
WO-1999055679-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 1999-11-04 WO disclosed