SCHEMBL7792654

SCHEMBL7792654

COc1ccc(CCN)cc1.O=Cc1ccc(Oc2ccccc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.58
MAOB P27338 5/20 0.54
ALDH1A1 P00352 2/20 0.53
CYP2A6 P11509 1/20 0.53
LTA4H P09960 2/20 0.50
KDM4E B2RXH2 1/20 0.47
HTT P42858 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
TTR P02766 1/20 0.47
FFAR1 O14842 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzaldehyde SCHEMBL7798573 0.91 TAAR1 (0.66) TAAR1MAOBALDH1A1CYP2A6LTA4H
SCHEMBL7792570 0.90 NPC1 (0.59) TAAR1MAOBALDH1A1LTA4HKDM4E
SCHEMBL7792264 0.89 ALDH1A1 (0.56) MAOBALDH1A1CYP2A6LTA4HKDM4E
SCHEMBL7800110 0.81 TAAR1 (0.60) TAAR1ALDH1A1CYP2A6KDM4ETTR
SCHEMBL5604883 0.80 ALDH1A1 (0.76) TAAR1MAOBALDH1A1CYP2A6LTA4H
Phenethylamine SCHEMBL22129843 0.80 TAAR1 (0.84) TAAR1MAOBCYP2A6LTA4HSMN1; SMN2
SCHEMBL740325 0.80 HTR2A (0.62) TAAR1CYP2A6LTA4HSMN1; SMN2FFAR1
SCHEMBL28527968 0.80 HTR2A (0.62) TAAR1CYP2A6LTA4HSMN1; SMN2FFAR1
Anisaldehyde SCHEMBL6814373 0.80 ALDH1A1 (0.83) ALDH1A1CYP2A6LTA4HNPC1RAB9A
SCHEMBL7798169 0.80 NPC1 (0.63) MAOBALDH1A1CYP2A6LTA4HKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1076649-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 2001-02-21 EP disclosed
US-6127381-A A MELANOCORTIN RECEPTOR LIGAND FOR REGULATING FOOD INTAKE AND BODY WEIGHT, REGULATING CYTOKINE ACTIVITY, ANTI-INFLAMMATORY ACTIVITY LION BIOSCIENCE AG (DE) 2000-10-03 US disclosed
WO-1999055679-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 1999-11-04 WO disclosed