SCHEMBL7792570

SCHEMBL7792570

COc1ccc(CCN)cc1.O=Cc1cccc(Oc2ccccc2)c1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.59
RAB9A P51151 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
TAAR1 Q96RJ0 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.52
KDM4E B2RXH2 1/20 0.52
ALDH1A1 P00352 1/20 0.52
HTT P42858 1/20 0.52
MAOB P27338 7/20 0.49
MAOA P21397 2/20 0.47
TTR P02766 1/20 0.46
LTA4H P09960 1/20 0.45
LPAR1 Q92633 1/20 0.43
LPAR5 Q9H1C0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7798169 0.91 NPC1 (0.63) NPC1RAB9ATDP1SMN1; SMN2KDM4E
SCHEMBL7792654 0.90 TAAR1 (0.58) NPC1RAB9ATDP1TAAR1SMN1; SMN2
Benzaldehyde SCHEMBL7798573 0.87 TAAR1 (0.66) NPC1RAB9ATDP1TAAR1ALDH1A1
SCHEMBL273688 0.84 NPC1 (0.65) NPC1RAB9ATDP1SMN1; SMN2KDM4E
SCHEMBL30866102 0.84 NPC1 (0.65) NPC1RAB9ATDP1SMN1; SMN2KDM4E
Glycine SCHEMBL8204567 0.83 NPC1 (0.56) NPC1RAB9ATDP1SMN1; SMN2KDM4E
SCHEMBL7792557 0.82 MAOB (0.52) NPC1RAB9ATDP1TAAR1SMN1; SMN2
SCHEMBL7798052 0.81 TAAR1 (0.56) TAAR1KDM4EALDH1A1MAOBMAOA
SCHEMBL7792264 0.81 ALDH1A1 (0.56) NPC1RAB9ATDP1SMN1; SMN2KDM4E
Benzaldehyde SCHEMBL14677731 0.80 TAAR1 (0.71) NPC1RAB9ATDP1TAAR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1076649-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 2001-02-21 EP disclosed
US-6127381-A A MELANOCORTIN RECEPTOR LIGAND FOR REGULATING FOOD INTAKE AND BODY WEIGHT, REGULATING CYTOKINE ACTIVITY, ANTI-INFLAMMATORY ACTIVITY LION BIOSCIENCE AG (DE) 2000-10-03 US disclosed
WO-1999055679-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 1999-11-04 WO disclosed