SCHEMBL7792549

SCHEMBL7792549

Cc1c(C)c(OCc2ccccc2)c(CC(=O)Cc2ccc(OCc3ccccc3)cc2OCc2ccccc2)c(C)c1OCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.43
MAOB P27338 4/20 0.43
S1PR1 P21453 1/20 0.42
S1PR5 Q9H228 1/20 0.42
PPARA Q07869 1/20 0.41
PTPN1 P18031 1/20 0.40
ALOX5 P09917 1/20 0.40
ACHE P22303 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
SRD5A2 P31213 1/20 0.40
HSD17B10 Q99714 1/20 0.40
NR4A2 P43354 2/20 0.40
CASP3 P42574 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8060518 0.95 L3MBTL1 (0.46) L3MBTL1MAOBPPARAMTNR1AMTNR1B
SCHEMBL7792657 0.95 L3MBTL1 (0.46) L3MBTL1MAOBPPARAMTNR1AMTNR1B
SCHEMBL7796504 0.81 MAOB (0.37) L3MBTL1MAOBS1PR1S1PR5PPARA
SCHEMBL3813849 0.78 PTGER1 (0.54) L3MBTL1MAOBALOX5KDM4EALDH1A1
SCHEMBL7792552 0.77 FFAR1 (0.47) L3MBTL1MAOBS1PR1S1PR5PPARA
SCHEMBL7795041 0.76 ABCB1 (0.45) MAOBKDM4EALDH1A1HPGDMTNR1A
SCHEMBL5446276 0.76 L3MBTL1 (0.53) L3MBTL1MAOBPPARAALOX5ALDH1A1
SCHEMBL9840655 0.76 L3MBTL1 (0.49) L3MBTL1MAOBS1PR1S1PR5ALOX5
SCHEMBL3023243 0.75 MAOB (0.51) L3MBTL1MAOBPPARAALOX5CYP1A2
SCHEMBL8060522 0.74 FFAR1 (0.49) L3MBTL1MAOBPPARAMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0909267-B1 NOVEL 1,3-DIPHENYLPROPANE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST TYROSINASE AND PROCESS FOR PREPARATION THEREOF LG CHEMICAL LTD (KR) 2001-11-21 EP disclosed
US-6093836-A INHIBITORY ACTIVITY AGAINT MELANIN BIOSYNTHESIS; WHITENING SUBSTANCES FOR MEDICAMENTS, COSMETICS LG CHEMICAL LTD. (KR) 2000-07-25 US disclosed
EP-0909267-A1 NOVEL 1,3-DIPHENYLPROPANE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST TYROSINASE AND PROCESS FOR PREPARATION THEREOF LG CHEMICAL LIMITED (KR) 1999-04-21 EP disclosed
WO-1998039279-A1 NOVEL 1,3-DIPHENYLPROPANE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST TYROSINASE AND PROCESS FOR PREPARATION THEREOF LG CHEMICAL LTD. (KR) 1998-09-11 WO disclosed