SCHEMBL7792800

SCHEMBL7792800

N#CC(CCC(=O)O)(CCC(=O)O)c1ccc(OC(F)F)c(OC(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.42
HSD17B10 Q99714 1/20 0.42
PDE4A P27815 11/20 0.41
PDE4B Q07343 4/20 0.41
PDE4C Q08493 4/20 0.41
PDE4D Q08499 4/20 0.41
FFAR1 O14842 2/20 0.41
CYP2C9 P11712 1/20 0.39
KCNH2 Q12809 1/20 0.39
CACNA1C Q13936 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.35
STING1 Q86WV6 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ESR1 P03372 1/20 0.33
CYP3A4 P08684 1/20 0.33
ESR2 Q92731 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7421932 0.93 CASP1 (0.53) CASP1HSD17B10PDE4APDE4BPDE4C
SCHEMBL7532617 0.88 PDE4D (0.51) PDE4APDE4BPDE4CPDE4DKCNH2
SCHEMBL7866895 0.87 PDE4B (0.49) PDE4APDE4BPDE4CPDE4D
SCHEMBL7415171 0.86 HSD17B10 (0.45) CASP1HSD17B10PDE4APDE4BPDE4C
SCHEMBL7416817 0.82 HSD17B10 (0.52) CASP1HSD17B10FFAR1L3MBTL1CYP3A4
SCHEMBL7384417 0.80 HSD17B10 (0.66) CASP1HSD17B10L3MBTL1ALDH1A1CYP3A4
SCHEMBL8677454 0.80 PDE4D (0.46) PDE4APDE4BPDE4CPDE4DKCNH2
SCHEMBL8677452 0.77 PDE4D (0.45) PDE4APDE4BPDE4CPDE4DKCNH2
SCHEMBL7858805 0.76 PDE4D (0.48) CASP1HSD17B10PDE4APDE4BPDE4C
SCHEMBL7865357 0.76 PDE4B (0.52) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636026-B1 COMPOUNDS USEFUL FOR TREATING INFLAMMATORY DISEASES AND INHIBITING PRODUCTION OF TUMOR NECROSIS FACTOR SMITHKLINE BEECHAM CORP (US) 2001-12-05 EP disclosed
US-5605923-A Compounds useful for treating inflammatory diseases and inhibiting production of tumor necrosis factor SMITHKLINE BEECHAM CORPORATION (US) 1997-02-25 US disclosed