SCHEMBL7794611

SCHEMBL7794611

COc1cc2nc(N)nc(-c3ccccc3)c2c(O)c1OC

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.54
ADORA1 P30542 6/20 0.54
SLC10A2 Q12908 1/20 0.47
SMPD3 Q9NY59 3/20 0.44
NOX1 Q9Y5S8 1/20 0.44
NUDT1 P36639 1/20 0.43
DHFR P00374 1/20 0.43
TYMS P04818 1/20 0.43
WHR1 P49842 1/20 0.42
MAPT P10636 1/20 0.42
ADORA2B P29275 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27775603 0.81 SLC10A2 (0.46) ADORA2AADORA1SLC10A2DHFRMAPT
SCHEMBL7800633 0.80 ADORA2A (0.45) ADORA2AADORA1SLC10A2DHFR
SCHEMBL3778066 0.77 SLC10A2 (0.56) ADORA2AADORA1SLC10A2SMPD3NOX1
SCHEMBL27754823 0.75 SLC2A1 (0.46) ADORA2AADORA1SLC10A2DHFRMAPT
SCHEMBL27755188 0.75 SLC10A2 (0.56) ADORA2AADORA1SLC10A2DHFRMAPT
SCHEMBL1257435 0.75 WHR1 (0.71) ADORA2AADORA1NUDT1DHFRWHR1
SCHEMBL30759714 0.75 WHR1 (0.71) ADORA2AADORA1NUDT1DHFRWHR1
SCHEMBL27775599 0.75 ADORA2A (0.52) ADORA2AADORA1SLC10A2DHFRADORA2B
SCHEMBL27755284 0.75 EGFR (0.46) ADORA2AADORA1SLC10A2DHFR
SCHEMBL27754944 0.73 DHFR (0.45) ADORA2AADORA1SLC10A2DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2531487-A1 ARYL BENZYLAMINE COMPOUNDS Novartis AG (CH) 2012-12-12 EP disclosed
EP-1158968-A2 JAK-3 INHIBITORS FOR TREATING ALLERGIC DISORDERS Parker Hughes Institute (US) 2001-12-05 EP disclosed
WO-2000051587-A2 JAK-3 INHIBITORS FOR TREATING ALLERGIC DISORDERS PARKER HUGHES INSTITUTE (US) 2000-09-08 WO disclosed