SCHEMBL7795312

SCHEMBL7795312

COC(=O)CCCC#CBr

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.56
LMNA P02545 3/20 0.41
ALDH1A1 P00352 2/20 0.41
CA12 O43570 3/20 0.41
CA14 Q9ULX7 3/20 0.41
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
PPARG P37231 3/20 0.37
PPARA Q07869 3/20 0.37
KDM4E B2RXH2 1/20 0.36
RECQL P46063 1/20 0.36
GLA P06280 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28035577 0.92 TSHR (0.52) TSHRLMNAALDH1A1CA12CA14
SCHEMBL2595476 0.92 TSHR (0.52) TSHRLMNAALDH1A1CA12CA14
SCHEMBL317846 0.82 TSHR (0.54) TSHRLMNAALDH1A1CA12CA14
SCHEMBL5250835 0.81 TSHR (0.58) TSHRLMNAALDH1A1CA12CA14
SCHEMBL18191271 0.81 TSHR (0.58) TSHRLMNAALDH1A1CA12CA14
SCHEMBL14198598 0.80 TSHR (0.52) TSHRLMNAALDH1A1KMT2AMEN1
SCHEMBL7966127 0.79 TSHR (0.56) TSHRALDH1A1CA12CA14KMT2A
SCHEMBL659218 0.79 TSHR (0.56) TSHRLMNAALDH1A1CA12CA14
SCHEMBL16288751 0.79 TSHR (0.56) TSHRLMNAALDH1A1CA12CA14
SCHEMBL7551344 0.79 TSHR (0.56) TSHRLMNAALDH1A1CA12CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103664605-B The preparation method of bromo-5,7, the 15-tri-alkynes-17-alkene stearic acid esters of bromination yne compounds E-18- SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2015-12-09 CN disclosed
WO-2014040477-A1 PROCESS FOR PREPARING BROMINATED ENYNE COMPOUND E-18-BROMO-5,7,15-TRIYNE-17-ENE OCTADECANOIC ACID ESTER 中国科学院上海药物研究所 (CN) 2014-03-20 WO disclosed
US-6310257-B2 ACIDOLYSIS OF EPOXIDE COMPOUND TO FORM CYCLOPENTENE DERIVATIVE NISSAN CHEMICAL INDUSTRIES, LTD (JP) 2001-10-30 US disclosed
US-20010012907-A1 Substituted cyclopentene derivatives and method for preparing the same NISSAN CHEMICAL INDUSTRIES, LTD. 2001-08-09 US disclosed
US-6191291-B1 OXIDATION OF A SUBSTITUTED CYCLOPENTADIENE DERIVATIVE WITH AN OXIDIZING AGENT TO FORM OXIRANE RING CONTAINING SUBSTITUTED CYCLOPENTADIENE DERIVATIVE NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2001-02-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010012907-A1 Substituted cyclopentene derivatives and method for preparing the same ACOX3, ACOX1, CBR1 TSHR 2128/4885LMNA 1107/4885ALDH1A1 448/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.