SCHEMBL7795660

SCHEMBL7795660

CCOc1cc(OC)c2c(c1)C(=O)c1cccc(OCCN3CCOCC3)c1-2

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
HTT P42858 1/20 0.47
CYP2D6 P10635 1/20 0.47
TSHR P16473 1/20 0.47
CHEK1 O14757 1/20 0.46
HTR2C P28335 2/20 0.46
HTR2B P41595 2/20 0.46
PTPN1 P18031 1/20 0.45
SYK P43405 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
BRD4 O60885 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27514211 0.96 ALDH1A1 (0.44) KDM4EALDH1A1HTTCYP2D6TSHR
SCHEMBL7796485 0.95 TSHR (0.49) KDM4EALDH1A1CYP2D6TSHRCHEK1
SCHEMBL7792104 0.95 KDM4E (0.50) KDM4EALDH1A1HTTCHEK1BRD4
SCHEMBL7786514 0.93 TSHR (0.46) KDM4EALDH1A1CYP2D6TSHRCHEK1
SCHEMBL7792479 0.93 CHEK1 (0.49) KDM4EALDH1A1HTTCYP2D6TSHR
SCHEMBL7792180 0.93 KDM4E (0.48) KDM4EALDH1A1HTTCHEK1BRD4
SCHEMBL7792176 0.93 KDM4E (0.50) KDM4EALDH1A1HTTTSHRBRD4
SCHEMBL7791821 0.93 CHEK1 (0.50) KDM4EALDH1A1CYP2D6TSHRCHEK1
Hydrochloric Acid SCHEMBL7792093 0.92 ALDH1A1 (0.45) KDM4EALDH1A1CYP2D6TSHRCHEK1
SCHEMBL7786319 0.91 POLB (0.50) KDM4EALDH1A1HTTTSHRHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906268-B1 ALKYLOXYAMINO SUBSTITUTED FLUORENONES AND THEIR USE AS PROTEIN KINASE C INHIBITORS AVENTIS PHARMA INC (US) 2001-11-28 EP disclosed
US-6004959-A HYPOTENSIVE, ANTITUMOR, ANTIINFLAMMATORY AND ANTIASTHMATIC AGENTS; ANGIOGENESIS AND ALVEOLAR MACROPHAGE ACTIVATION INHIBITORS HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US disclosed