SCHEMBL7795894

SCHEMBL7795894

FC(F)(F)c1cc2nc(S)[nH]c2cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 4/20 0.44
EGLN1 Q9GZT9 2/20 0.41
AR P10275 5/20 0.39
CACNA1G O43497 1/20 0.39
CACNA1C Q13936 1/20 0.39
GAA P10253 1/20 0.37
HTT P42858 1/20 0.37
NPY5R Q15761 1/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
NOTUM Q6P988 1/20 0.35
TRPA1 O75762 1/20 0.35
TRPM8 Q7Z2W7 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
CHEK2 O96017 1/20 0.34
RHEB Q15382 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7795887 0.93 EGLN1 (0.47) CACNA1HEGLN1ARCACNA1GCACNA1C
SCHEMBL2418527 0.83 CACNA1H (0.46) CACNA1HEGLN1ARCACNA1GCACNA1C
SCHEMBL10847054 0.81 AR (0.50) CACNA1HEGLN1ARCACNA1GGAA
SCHEMBL9814439 0.81 KDM4E (0.54) CACNA1HEGLN1ARCACNA1GCACNA1C
SCHEMBL12020706 0.80 MAPT (0.57) CACNA1HEGLN1ARCACNA1GCACNA1C
SCHEMBL5681325 0.80 HTR3E (0.49) CACNA1HEGLN1ARCACNA1GCACNA1C
SCHEMBL21066380 0.80 EGLN1 (0.44) CACNA1HEGLN1ARCACNA1GCACNA1C
SCHEMBL2105304 0.80 GAA (0.53) CACNA1HEGLN1ARCACNA1GGAA
SCHEMBL18659704 0.78 AR (0.50) CACNA1HEGLN1ARCACNA1GCACNA1C
SCHEMBL211043 0.77 ALDH1A1 (0.44) CACNA1HEGLN1ARCACNA1GGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0742210-B1 2-MERCAPTOBENZIMIDAZOLE DERIVATIVE AND ANTIHYPERLIPEMIC OR ANTIARTERIOSCLEROTIC AGENT CONTAINING THE SAME FUJI PHOTO FILM CO LTD (JP) 2001-11-21 EP disclosed
US-6288236-B1 PREVENTIVE AND THERAPEUTIC MEDICAMENT FOR HYPERLIPEMIA OR ARTERIAL SCLEROSIS. FUJI PHOTO FILM CO., LTD. (JP) 2001-09-11 US disclosed
US-6174907-B1 THERAPY AND PROPHYLAXIS OF HYPERLIPEMIA OR ARTERIAL SCLEROSIS; AS ADDITIVE OF A SILVER HALIDE PHOTOSENSITIVE MATERIAL, LIQUID CRYSTAL MATERIAL FUJI PHOTO FILM CO., LTD. (JP) 2001-01-16 US disclosed
US-5998456-A ANTILIPEMIC AGENTS FUJI PHOTO FILM CO., LTD. (JP) 1999-12-07 US disclosed
US-5962493-A HYPOLIPEMIC AGENTS; ANTICHOLESTEROL AGENTS FUJI PHOTO FILM CO., LTD. (JP) 1999-10-05 US disclosed
EP-0849259-A1 BENZIMIDAZOLE COMPOUNDS FUJI PHOTO FILM CO., LTD. (JP) 1998-06-24 EP disclosed
EP-0742210-A1 2-MERCAPTOBENZIMIDAZOLE DERIVATIVE AND ANTIHYPERLIPEMIC OR ANTIARTERIOSCLEROTIC AGENT CONTAINING THE SAME FUJI PHOTO FILM CO., LTD. (JP) 1996-11-13 EP disclosed