SCHEMBL7796711

SCHEMBL7796711

NC1=NC2(CCN(C(=O)c3ccc(N)cc3)CC2)Nc2ccccc21

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 10/20 0.58
NOS1 P29475 7/20 0.58
NEK2 P51955 1/20 0.47
NOS3 P29474 2/20 0.44
KCNH2 Q12809 1/20 0.43
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
CRBN Q96SW2 1/20 0.40
IP6K1 Q92551 2/20 0.39
IP6K3 Q96PC2 1/20 0.39
IP6K2 Q9UHH9 1/20 0.39
SCN5A Q14524 1/20 0.39
SCN9A Q15858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8379932 0.99 NOS2 (0.57) NOS2NOS1NEK2NOS3KCNH2
SCHEMBL7804452 0.93 NOS2 (0.57) NOS2NOS1NEK2NOS3CRBN
SCHEMBL7931778 0.92 NOS2 (0.57) NOS2NOS1NEK2NOS3KCNH2
SCHEMBL7796668 0.92 NOS2 (0.57) NOS2NOS1NEK2NOS3KCNH2
Hydrochloric Acid SCHEMBL8378262 0.92 NOS2 (0.56) NOS2NOS1NEK2NOS3KCNH2
Hydrochloric Acid SCHEMBL8376965 0.91 NOS2 (0.56) NOS2NOS1NEK2NOS3KCNH2
Hydrochloric Acid SCHEMBL8377866 0.91 NOS2 (0.56) NOS2NOS1NEK2NOS3KCNH2
SCHEMBL7804492 0.91 NOS2 (0.56) NOS2NOS1NEK2NOS3KCNH2
SCHEMBL7802943 0.91 NOS2 (0.61) NOS2NOS1NEK2NOS3KCNH2
SCHEMBL7806816 0.91 NOS2 (0.56) NOS2NOS1NEK2NOS3SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248745-B1 MIXTURE COMPRISING A CYCLOOXYGENASE-2 (COX-2) INHIBITOR AND A 1,2-DIHYDRO-4-AMINOQUINAZOLINE DERIVATIVE INHIBITOR OF INDUCED NITRIC OXIDE SYNTHASE (INOS); NON-STEROIDAL ANTIINFLAMMATORY AGENTS ASTRAZENECA AB (SE) 2001-06-19 US claimed
EP-1100505-A1 A PHARMACEUTICAL COMBINATION COMPRISING A COX-2 INHIBITOR AND A iNOS INHIBITOR AstraZeneca AB (SE) 2001-05-23 EP claimed
WO-2000000200-A1 A PHARMACEUTICAL COMBINATION COMPRISING A COX-2 INHIBITOR AND A iNOS INHIBITOR ASTRAZENECA AB (SE) 2000-01-06 WO claimed