SCHEMBL7931778

SCHEMBL7931778

NC1=NC2(CCN(C(=O)c3ccc(O)cc3)CC2)Nc2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 10/20 0.57
NOS1 P29475 7/20 0.57
NEK2 P51955 1/20 0.47
NOS3 P29474 2/20 0.44
KCNH2 Q12809 1/20 0.42
CRBN Q96SW2 1/20 0.39
IP6K1 Q92551 2/20 0.38
IP6K3 Q96PC2 1/20 0.38
IP6K2 Q9UHH9 1/20 0.38
USP2 O75604 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38
DHFR P00374 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8376965 0.99 NOS2 (0.56) NOS2NOS1NEK2NOS3KCNH2
SCHEMBL7796711 0.92 NOS2 (0.58) NOS2NOS1NEK2NOS3KCNH2
SCHEMBL7804452 0.92 NOS2 (0.57) NOS2NOS1NEK2NOS3CRBN
SCHEMBL7796668 0.91 NOS2 (0.57) NOS2NOS1NEK2NOS3KCNH2
Hydrochloric Acid SCHEMBL8379932 0.91 NOS2 (0.57) NOS2NOS1NEK2NOS3KCNH2
Hydrochloric Acid SCHEMBL8378262 0.91 NOS2 (0.56) NOS2NOS1NEK2NOS3KCNH2
Hydrochloric Acid SCHEMBL8377866 0.90 NOS2 (0.56) NOS2NOS1NEK2NOS3KCNH2
SCHEMBL7806816 0.90 NOS2 (0.56) NOS2NOS1NEK2NOS3ALDH1A1
SCHEMBL7943019 0.90 NEK2 (0.59) NOS2NOS1NEK2NOS3KCNH2
SCHEMBL7802943 0.90 NOS2 (0.61) NOS2NOS1NEK2NOS3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248745-B1 MIXTURE COMPRISING A CYCLOOXYGENASE-2 (COX-2) INHIBITOR AND A 1,2-DIHYDRO-4-AMINOQUINAZOLINE DERIVATIVE INHIBITOR OF INDUCED NITRIC OXIDE SYNTHASE (INOS); NON-STEROIDAL ANTIINFLAMMATORY AGENTS ASTRAZENECA AB (SE) 2001-06-19 US claimed