SCHEMBL7798052

SCHEMBL7798052

COc1ccccc1CCN.O=Cc1cccc(Oc2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.56
HRH1 P35367 1/20 0.54
TTR P02766 1/20 0.51
ALDH1A1 P00352 2/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
KDM4E B2RXH2 1/20 0.51
BACE1 P56817 1/20 0.45
POLB P06746 1/20 0.44
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
ADRA1A P35348 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7800110 0.89 TAAR1 (0.60) TAAR1HRH1TTRALDH1A1MEN1
SCHEMBL7792570 0.81 NPC1 (0.59) TAAR1TTRALDH1A1KDM4EMAOA
SCHEMBL7802655 0.78 MAOA (0.46) TTRALDH1A1MEN1KMT2AKDM4E
SCHEMBL25809767 0.77 HRH1 (0.58) TAAR1HRH1ADRA1A
SCHEMBL7798169 0.77 NPC1 (0.63) TTRALDH1A1KDM4EMAOAMAOB
SCHEMBL2075852 0.77 TTR (0.67) TTRALDH1A1MEN1KMT2APOLB
SCHEMBL2207553 0.77 NPC1 (0.64) ALDH1A1MEN1KMT2APOLBMAOA
SCHEMBL98478 0.77 MAOB (0.61) TTRALDH1A1MEN1KMT2AMAOA
SCHEMBL29484309 0.77 MAOB (0.61) TTRALDH1A1MEN1KMT2AMAOA
SCHEMBL11482497 0.77 MAOB (0.61) TTRALDH1A1MEN1KMT2AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1076649-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 2001-02-21 EP disclosed
US-6127381-A A MELANOCORTIN RECEPTOR LIGAND FOR REGULATING FOOD INTAKE AND BODY WEIGHT, REGULATING CYTOKINE ACTIVITY, ANTI-INFLAMMATORY ACTIVITY LION BIOSCIENCE AG (DE) 2000-10-03 US disclosed
WO-1999055679-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 1999-11-04 WO disclosed