SCHEMBL7798252

SCHEMBL7798252

Cc1ccc(C(F)[C](F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.41
ACHE P22303 4/20 0.40
KEAP1 Q14145 2/20 0.40
NFE2L2 Q16236 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
AGER Q15109 1/20 0.36
ALOX5 P09917 1/20 0.35
LMNA P02545 3/20 0.33
ALDH1A1 P00352 2/20 0.33
FFAR1 O14842 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
CA2 P00918 1/20 0.33
LPL P06858 1/20 0.33
LIPG Q9Y5X9 1/20 0.33
ORAI1 Q96D31 1/20 0.33
ORAI2 Q96SN7 1/20 0.33
ORAI3 Q9BRQ5 1/20 0.33
TRPV6 Q9H1D0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9953863 0.77 IDO1 (0.41) LMNAALDH1A1SMN1; SMN2CES2CES1
SCHEMBL2399005 0.76 KEAP1 (0.53) ACHEKEAP1NFE2L2ALOX5LMNA
SCHEMBL23554861 0.76 CYP3A4 (0.41) CHRNA7ACHEKEAP1NFE2L2TDP1
SCHEMBL28037840 0.74 ACHE (0.44) CHRNA7ACHEKEAP1NFE2L2TDP1
SCHEMBL371162 0.73 ACHE (0.50) CHRNA7ACHETDP1AGERALOX5
SCHEMBL2055581 0.73 ACHE (0.50) CHRNA7ACHETDP1AGERALOX5
SCHEMBL11861772 0.72 KEAP1 (0.45) ACHEKEAP1NFE2L2TDP1ALOX5
SCHEMBL14417193 0.70 ACHE (0.47) CHRNA7ACHEKEAP1NFE2L2TDP1
SCHEMBL17020102 0.70 CHRNA7 (0.46) CHRNA7ACHEKEAP1NFE2L2TDP1
SCHEMBL9732281 0.70 CHRNA7 (0.46) CHRNA7ACHEKEAP1NFE2L2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1076649-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 2001-02-21 EP claimed
WO-1999055679-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 1999-11-04 WO claimed