SCHEMBL7799074

SCHEMBL7799074

C=CC(Cc1ccccc1)N(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.44
SLC6A2 P23975 3/20 0.43
SLC6A4 P31645 2/20 0.43
SLC6A3 Q01959 2/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
HTR2A P28223 1/20 0.43
ADRA1A P35348 1/20 0.43
OPRK1 P41145 1/20 0.43
KCNH2 Q12809 1/20 0.43
TSHR P16473 2/20 0.39
EPHX1 P07099 2/20 0.39
ALDH1A1 P00352 2/20 0.39
GAA P10253 2/20 0.38
KMT2A Q03164 2/20 0.38
HPGD P15428 1/20 0.38
NPBWR1 P48145 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MCHR1 Q99705 1/20 0.38
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2600695 1.00 SIGMAR1 (0.44) SIGMAR1SLC6A2SLC6A4SLC6A3ADRA2B
Hydrochloric Acid SCHEMBL7799087 0.98 SIGMAR1 (0.42) SIGMAR1SLC6A2SLC6A4SLC6A3ADRA2B
SCHEMBL7799023 0.86 L3MBTL1 (0.49) SIGMAR1TSHRALDH1A1
SCHEMBL9222606 0.83 TAAR1 (0.39) SIGMAR1SLC6A2SLC6A4SLC6A3ADRA2B
SCHEMBL8717938 0.81 SIGMAR1 (0.44) SIGMAR1SLC6A2SLC6A4SLC6A3ADRA2B
SCHEMBL475432 0.81 EPHX1 (0.44) SIGMAR1SLC6A2SLC6A4SLC6A3ADRA2B
SCHEMBL475431 0.81 EPHX1 (0.44) SIGMAR1SLC6A2SLC6A4SLC6A3ADRA2B
SCHEMBL18085369 0.80 TSHR (0.39) SIGMAR1SLC6A2SLC6A4SLC6A3ADRA2B
SCHEMBL151553 0.79 ALDH1A1 (0.43) SIGMAR1TSHRALDH1A1GAAKMT2A
SCHEMBL995542 0.78 SLC6A2 (0.44) SIGMAR1SLC6A2SLC6A4SLC6A3ADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0748801-B1 2-ISOXAZOLINE DERIVATIVE AND PROCESS FOR PRODUCING THE SAME, AND PROCESS FOR PRODUCING RELATED DERIVATIVES FROM THE SAME DAICEL CHEM (JP) 2001-12-19 EP disclosed
US-6018069-A 2-isoxazoline derivative and process for producing the same and process for producing related derivatives from the same DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 2000-01-25 US disclosed
US-5994558-A 2-isoxazoline derivative and process for producing the same; and process for producing related derivatives from the same DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1999-11-30 US disclosed
US-5962692-A 2-isoxazoline derivative and process for producing the same, and process for producing related derivatives from the same DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1999-10-05 US disclosed
US-5750717-A 2-isoxazoline derivative and process for producing the same, and process for producing related derivatives from the same DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-12 US disclosed
EP-0748801-A1 2-ISOXAZOLINE DERIVATIVE AND PROCESS FOR PRODUCING THE SAME, AND PROCESS FOR PRODUCING RELATED DERIVATIVES FROM THE SAME DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-18 EP disclosed