SCHEMBL7800097

SCHEMBL7800097

COc1cccc(CCN)c1.O=Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.61
KDM4E B2RXH2 2/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
MAOB P27338 4/20 0.47
CHRM2 P08172 3/20 0.45
CHRM1 P11229 3/20 0.45
CHRM3 P20309 3/20 0.45
AOC3 Q16853 1/20 0.43
ACHE P22303 2/20 0.42
ALDH1A1 P00352 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
IDO1 P14902 1/20 0.40
AGXT P21549 1/20 0.40
SIGMAR1 Q99720 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7800391 0.92 TAAR1 (0.59) TAAR1KDM4EMEN1KMT2AMAOB
Benzoic Acid SCHEMBL7800774 0.91 TAAR1 (0.50) TAAR1KDM4EMEN1KMT2AACHE
SCHEMBL7802621 0.90 MAOB (0.47) TAAR1KDM4EMEN1KMT2AMAOB
4-Methylbenzoic Acid SCHEMBL7792499 0.88 TAAR1 (0.47) TAAR1KDM4EMEN1KMT2AMAOB
SCHEMBL8035116 0.87 PTGES (0.48) TAAR1KDM4EMEN1KMT2AMAOB
SCHEMBL7798027 0.87 KDM4E (0.46) TAAR1KDM4EMEN1KMT2AMAOB
SCHEMBL7801502 0.86 TAAR1 (0.55) TAAR1MEN1KMT2AMAOBALDH1A1
Benzoic Acid SCHEMBL7800370 0.83 MEN1 (0.53) TAAR1KDM4EMEN1KMT2AMAOB
Benzaldehyde SCHEMBL14677731 0.82 TAAR1 (0.71) TAAR1KDM4EMEN1KMT2AMAOB
Phenethylamine SCHEMBL7801605 0.82 TAAR1 (0.53) TAAR1MAOBIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1076649-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 2001-02-21 EP disclosed
US-6127381-A A MELANOCORTIN RECEPTOR LIGAND FOR REGULATING FOOD INTAKE AND BODY WEIGHT, REGULATING CYTOKINE ACTIVITY, ANTI-INFLAMMATORY ACTIVITY LION BIOSCIENCE AG (DE) 2000-10-03 US disclosed
WO-1999055679-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 1999-11-04 WO disclosed