SCHEMBL7800958

SCHEMBL7800958

CC(C)CCN(C(=O)O)C(=O)N(CCc1ccccc1)CC(=O)C(C)(C)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.41
OPRD1 P41143 2/20 0.41
OPRK1 P41145 2/20 0.41
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
LMNA P02545 1/20 0.39
PKM P14618 1/20 0.39
MEN1 O00255 5/20 0.39
KMT2A Q03164 5/20 0.39
AOC3 Q16853 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
TSHR P16473 1/20 0.37
KDM4E B2RXH2 1/20 0.37
RCE1 Q9Y256 1/20 0.36
HTT P42858 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7798540 0.73 OPRM1 (0.39) OPRM1OPRD1OPRK1HDAC1HDAC6
SCHEMBL28466070 0.69 HDAC1 (0.51) HDAC1HDAC6MEN1KMT2AL3MBTL1
SCHEMBL13434109 0.69 SMN1; SMN2 (0.48) OPRM1OPRD1OPRK1HDAC1HDAC6
SCHEMBL27460199 0.68 MEN1 (0.42) HDAC1HDAC6MEN1KMT2AAOC3
Bicarbonate SCHEMBL27892668 0.68 TSHR (0.59) LMNAPKMMEN1KMT2ANPC1
SCHEMBL9823156 0.67 HDAC1 (0.54) HDAC1HDAC6LMNAMEN1KMT2A
SCHEMBL8577651 0.67 MEN1 (0.39) OPRM1OPRD1OPRK1LMNAPKM
SCHEMBL8502790 0.67 MEN1 (0.44) OPRM1OPRD1OPRK1LMNAPKM
SCHEMBL8504370 0.67 AOC3 (0.42) OPRM1OPRD1OPRK1LMNAPKM
SCHEMBL3050230 0.66 MEN1 (0.46) HDAC1HDAC6LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159260-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000055124-A2 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed