SCHEMBL7798540

SCHEMBL7798540

CC(C)CCN(C(=O)OCc1ccccc1)C(=O)N(CCc1ccccc1)CC(O)C(C)(C)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.39
OPRD1 P41143 2/20 0.39
OPRK1 P41145 2/20 0.39
ABCB1 P08183 1/20 0.37
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
KDM4E B2RXH2 1/20 0.36
CCR6 P51684 1/20 0.35
PAX8 Q06710 1/20 0.35
MMP8 P22894 1/20 0.35
MMP14 P50281 1/20 0.35
LMNA P02545 1/20 0.35
PKM P14618 1/20 0.35
CTSK P43235 2/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
ALDH1A1 P00352 1/20 0.35
AOC3 Q16853 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7790158 0.78 CCR6 (0.42) OPRM1OPRD1OPRK1CCR6PAX8
SCHEMBL6181959 0.74 CTSL (0.40) OPRM1OPRD1OPRK1CCR6PAX8
SCHEMBL7799705 0.74 CCR6 (0.38) OPRM1OPRD1OPRK1ABCB1CCR6
SCHEMBL7800958 0.73 OPRM1 (0.41) OPRM1OPRD1OPRK1HDAC1HDAC6
SCHEMBL6183141 0.73 ALOX5 (0.43) ABCB1CCR6PAX8CTSKCTSL
SCHEMBL6183149 0.72 CTSS (0.44) CTSKCTSLCTSBCTSSALDH1A1
SCHEMBL7137505 0.71 SMN1; SMN2 (0.41) CTSKCTSLCTSB
SCHEMBL6183588 0.70 CTSS (0.43) CCR6PAX8CTSKCTSLCTSB
SCHEMBL6183195 0.70 CTSS (0.42) CTSKCTSLCTSBCTSSALDH1A1
SCHEMBL12130679 0.70 KMT2A (0.50) ABCB1CCR6PAX8LMNACTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159260-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000055124-A2 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed