SCHEMBL7801013

SCHEMBL7801013

CCCCS(=O)(=O)Nc1ccc(Cl)c(C(=O)OC(C)=O)c1Cl.O=C(O)C[C@H](NC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 13/20 0.46
CASP3 P42574 4/20 0.41
SIRT2 Q8IXJ6 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
CTSL P07711 1/20 0.39
CTSS P25774 1/20 0.39
MME P08473 1/20 0.37
ECE1 P42892 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6802229 0.91 CASP1 (0.46) CASP1CASP3SIRT2SIRT1CTSL
SCHEMBL6798489 0.80 CASP1 (0.47) CASP1CASP3MMEECE1
SCHEMBL7179653 0.73 CASP1 (0.49) CASP1CASP3MMEECE1
SCHEMBL6797163 0.73 CASP3 (0.50) CASP1CASP3MMEECE1
SCHEMBL6800922 0.72 CASP1 (0.43) CASP1CASP3
SCHEMBL14989128 0.71 CASP1 (0.57) CASP1SIRT2SIRT1CTSLCTSS
SCHEMBL376886 0.70 CASP1 (0.67) CASP1MMEECE1
SCHEMBL554032 0.70 CASP1 (0.67) CASP1MMEECE1
SCHEMBL613386 0.70 CASP1 (0.67) CASP1MMEECE1
SCHEMBL8511225 0.70 BRAF (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623592-B1 Peptide analogs as irreversible interleukin-1beta protease inhibitors VERTEX PHARMA (US) 2001-06-27 EP disclosed
EP-0623592-A1 Peptide analogs as irreversible interleukin-1beta protease inhibitors STERLING WINTHROP INC. (US) 1994-11-09 EP disclosed