SCHEMBL7801221

SCHEMBL7801221

CC(NC(c1ccc(F)cc1)c1ccccc1Nc1c(O)c(=O)c1=O)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 5/20 0.41
CXCR1 P25024 2/20 0.41
NPC1 O15118 1/20 0.39
MAPKAPK2 P49137 2/20 0.37
ALDH1A1 P00352 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
KDM4E B2RXH2 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
CCR6 P51684 1/20 0.36
TEAD4 Q15561 1/20 0.35
CXCL8 P10145 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7801287 0.99 CXCR2 (0.41) CXCR2CXCR1NPC1MAPKAPK2ALDH1A1
SCHEMBL7801983 0.92 CXCR2 (0.40) CXCR2CXCR1MAPKAPK2ALDH1A1CCR6
SCHEMBL7801434 0.92 CXCR2 (0.40) CXCR2CXCR1MAPKAPK2ALDH1A1CCR6
Hydrochloric Acid SCHEMBL7804257 0.91 CXCR2 (0.40) CXCR2CXCR1MAPKAPK2ALDH1A1CCR6
Hydrochloric Acid SCHEMBL7795500 0.90 ALDH1A1 (0.42) CXCR2CXCR1MAPKAPK2ALDH1A1CYP3A4
SCHEMBL7805393 0.89 CXCR2 (0.40) CXCR2CXCR1MAPKAPK2CCR6TEAD4
SCHEMBL7795412 0.89 CXCR2 (0.40) CXCR2CXCR1MAPKAPK2CCR6TEAD4
SCHEMBL7795443 0.89 CXCR2 (0.41) CXCR2CXCR1CYP3A4CYP2C9CCR6
SCHEMBL7804119 0.89 CXCR2 (0.41) CXCR2CXCR1CYP3A4CYP2C9CCR6
Hydrochloric Acid SCHEMBL7803652 0.89 CXCR2 (0.39) CXCR2CXCR1MAPKAPK2CCR6TEAD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP claimed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed