SCHEMBL7801541

SCHEMBL7801541

NCCc1ccc(Cl)cc1.O=Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.51
MAOB P27338 9/20 0.46
RHOC P08134 2/20 0.40
RHOA P61586 2/20 0.40
KCNH2 Q12809 1/20 0.40
TMEM97 Q5BJF2 1/20 0.40
CNR1 P21554 1/20 0.39
HSD17B10 Q99714 1/20 0.38
PNMT P11086 1/20 0.37
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzoic Acid SCHEMBL7798267 0.88 TAAR1 (0.40) TAAR1MAOBRHOCRHOA
Tyramine SCHEMBL8035697 0.86 TAAR1 (0.51) TAAR1MAOB
SCHEMBL7798427 0.85 SRD5A2 (0.40) TAAR1RHOCRHOALMNAPOLB
4-Methylbenzoic Acid SCHEMBL7792518 0.85 SCN5A (0.40) TAAR1RHOCRHOALMNAPOLB
Phenethylamine SCHEMBL7801605 0.85 TAAR1 (0.53) TAAR1MAOB
SCHEMBL7792354 0.85 TAAR1 (0.58) TAAR1MAOBRHOCRHOAPNMT
SCHEMBL7802656 0.84 RXRA (0.47) MAOBLMNAPOLBMAPT
SCHEMBL7801502 0.82 TAAR1 (0.55) TAAR1MAOB
SCHEMBL18002359 0.81 RHOC (0.43) RHOCRHOAKCNH2TMEM97CNR1
SCHEMBL7801557 0.80 MAOB (0.51) TAAR1MAOBLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1076649-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 2001-02-21 EP disclosed
US-6127381-A A MELANOCORTIN RECEPTOR LIGAND FOR REGULATING FOOD INTAKE AND BODY WEIGHT, REGULATING CYTOKINE ACTIVITY, ANTI-INFLAMMATORY ACTIVITY LION BIOSCIENCE AG (DE) 2000-10-03 US disclosed
WO-1999055679-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 1999-11-04 WO disclosed