SCHEMBL7803853

SCHEMBL7803853

CN(C)CCOc1cccc(N2CC(c3ccccc3)OC2=O)c1

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FADS1 O60427 6/20 0.55
GRM2 Q14416 8/20 0.49
HTR6 P50406 1/20 0.47
HSD11B1 P28845 2/20 0.47
HDAC6 Q9UBN7 1/20 0.44
ALOX5 P09917 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7944255 0.80 FADS1 (0.45) FADS1HTR6HSD11B1
SCHEMBL7805594 0.78 FADS1 (0.48) FADS1GRM2HTR6
SCHEMBL9016279 0.75 FADS1 (0.79) FADS1GRM2HTR6HSD11B1
SCHEMBL7770572 0.73 GRM2 (0.54) FADS1GRM2HTR6
SCHEMBL7776725 0.71 FADS1 (0.60) FADS1GRM2HTR6HSD11B1
SCHEMBL1268405 0.69 HTR6 (0.55) FADS1GRM2HTR6HSD11B1
SCHEMBL28023734 0.69 FADS1 (0.60) FADS1GRM2HTR6HSD11B1
SCHEMBL2830693 0.68 GRM2 (0.74) GRM2
SCHEMBL4953049 0.68 SLC8A1 (0.61)
SCHEMBL7775283 0.67 FADS1 (0.65) FADS1GRM2HTR6HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1071670-A1 NOVEL DIPHENYL-SUBSTITUTED 5-RING-HETEROCYCLES, METHOD FOR PRODUCING THEM AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM KG (DE) 2001-01-31 EP disclosed
WO-1999054314-A1 NOVEL DIPHENYL-SUBSTITUTED 5-RING-HETEROCYCLES, METHOD FOR PRODUCING THEM AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-10-28 WO disclosed