SCHEMBL7804133

SCHEMBL7804133

CCOC(=O)CC(Cc1ccc(O)cc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.48
ESR2 Q92731 6/20 0.48
PPARG P37231 4/20 0.46
FFAR1 O14842 3/20 0.45
EPHX2 P34913 1/20 0.45
F2 P00734 2/20 0.45
F10 P00742 1/20 0.45
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
HSP90AA1 P07900 1/20 0.42
MAPT P10636 1/20 0.42
CRHBP P24387 1/20 0.42
KMT2A Q03164 1/20 0.42
CRHR2 Q13324 1/20 0.42
TRPM2 O94759 1/20 0.41
SLC6A9 P48067 1/20 0.41
MTOR P42345 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8371455 0.90 PPARG (0.45) PPARGFFAR1EPHX2F2F10
SCHEMBL9857070 0.89 SLC6A9 (0.52) PPARGFFAR1EPHX2F2F10
SCHEMBL7797631 0.88 THRB (0.50) PPARGFFAR1EPHX2F2F10
SCHEMBL27535203 0.84 ESR1 (0.51) ESR1ESR2F2F10KDM4E
SCHEMBL8329187 0.83 F2 (0.55) ESR1ESR2F2F10
SCHEMBL13236836 0.83 FFAR1 (0.46) PPARGFFAR1KDM4EMEN1HSP90AA1
SCHEMBL6490172 0.82 ESR1 (0.49) ESR1ESR2PPARGFFAR1SLC6A9
SCHEMBL6533433 0.77 F10 (0.47) ESR1ESR2FFAR1F2F10
SCHEMBL6533437 0.77 F10 (0.47) ESR1ESR2FFAR1F2F10
SCHEMBL15687505 0.77 ESR1 (0.50) ESR1ESR2FFAR1F2F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1236767-C Vitronectin receptor antagonists SMITHKLINE BEECHAM CORP (US) 2006-01-18 CN disclosed
US-6881736-B1 Vitronectin receptor antagonists SMITHKLINE BEECHAM CORPORATION (US) 2005-04-19 US disclosed
US-6881736-B1 Vitronectin receptor antagonists SMITHKLINE BEECHAM CORPORATION (US) 2005-04-19 US disclosed
CN-1377269-A Vitronectin receptor antagonists SMITHKLINE BEECHAM CORP (US) 2002-10-30 CN disclosed