SCHEMBL7804895

SCHEMBL7804895

Nc1c(Cl)cc(-c2nn(C3CC4CCC(C3)N4CCc3ccccc3)c(=O)o2)c2c1OCCO2

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 8/20 0.42
HRH3 Q9Y5N1 1/20 0.37
CHRNA7 P36544 3/20 0.37
OPRM1 P35372 3/20 0.35
OPRD1 P41143 3/20 0.35
OPRK1 P41145 1/20 0.35
KCNH2 Q12809 1/20 0.35
GPR55 Q9Y2T6 1/20 0.34
CNR1 P21554 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Capeserod SCHEMBL4707724 0.87 HTR4 (0.45) HTR4GPR55CNR1
Capeserod SCHEMBL399091 0.86 HTR4 (0.44) HTR4GPR55CNR1
SCHEMBL7810023 0.86 CHRNA7 (0.38) HRH3CHRNA7OPRM1OPRD1OPRK1
SCHEMBL7799598 0.85 HTR4 (0.44) HTR4
Bromide SCHEMBL7946667 0.84 HTR4 (0.43) HTR4
SCHEMBL7810030 0.83 HRH3 (0.37) HRH3CHRNA7OPRM1OPRD1OPRK1
Hydrochloric Acid SCHEMBL7946706 0.82 CHRNA7 (0.36) HRH3CHRNA7OPRM1OPRD1OPRK1
SCHEMBL7804890 0.78 HTR4 (0.46) HTR4
Hydrochloric Acid SCHEMBL7945299 0.77 HTR4 (0.46) HTR4
SCHEMBL8303718 0.77 HTR4 (0.52) HTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0975631-B1 5-ARYL-3-(8-AZABICYCLO[3.2.1]OCT-3-YL)-1,3,4-OXADIAZOL-2(3H)-ONE DERIVATIVES AS 5-HT4 RECEPTOR LIGANDS SANOFI SYNTHELABO (FR) 2001-10-04 EP disclosed
US-6255319-B1 ANTISEROTONIN AGENT SANOFI-SYNTHELABO (FR) 2001-07-03 US disclosed